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Search Results for " aha1 "
Targets Recommended: Others

3

抑制剂 & 化合物

1

重组蛋白

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Cat. No. Product Name Target Signaling Pathways
T62307 Aha1/Hsp90-IN-1

Others Others
Aha1/Hsp90-IN-1 (Compound 17) 是一种 Aha1/Hsp90 complex 抑制剂,对 tau 蛋白聚集具有抑制作用。Aha1/Hsp90-IN-1 能够破坏 Aha1/Hsp90 的相互作用 (IC50: 3.32 μM)。
T69571 SEW84

Others Others
SEW84 是 Aha1 刺激的 Hsp90(ASH) ATP 酶活性的抑制剂。SEW84 抑制 Aha1 刺激的 Hsp90(ASH) 活性,IC50值为 0.3 μM。SEW84 可用于蛋白质沉积疾病的研究。
T63273 KU-177

Others Others
KU-177 是一种有效的 Hsp90ATP 酶同系物 1 (Aha1) 抑制剂,能够消融 Aha1 驱动的 Hsp90 依赖性 tau 聚集增强。KU-177 能够阻碍 Aha1/Hsp90 相互作用,其IC50 值为 4.08 μM,但对Hsp90的再折叠荧光素酶的能力不造成影响。KU-177 可以阻碍癌细胞生长,诱导其凋亡 (apoptosis),能够用于研究 Tau 病。

化合物

Aha1/Hsp90-IN-1
Cat.No: T62307
Synonym:
Target: Others
SEW84
Cat.No: T69571
Synonym:
Target: Others
KU-177
Cat.No: T63273
Synonym:
Target: Others
Cat. No. Product Name Species Expression System
TMPH-00887 AHSA1 Protein, Human, Recombinant (GST)

C14orf3,p38,Activator of 90 kDa heat shock protein ...

Human E. coli
Acts as a co-chaperone of HSP90AA1. Activates the ATPase activity of HSP90AA1 leading to increase in its chaperone activity. Competes with the inhibitory co-chaperone FNIP1 for binding to HSP90AA1, thereby providing a reciprocal regulatory mechanism for chaperoning of client proteins. Competes with the inhibitory co-chaperone TSC1 for binding to HSP90AA1, thereby providing a reciprocal regulatory mechanism for chaperoning of client proteins. AHSA1 Protein, Human, Recombinant (GST) is expressed i...

重组蛋白

AHSA1 Protein, Human, Recombinant (GST)
Cat.No: TMPH-00887
Species: Human
Expression System: E. coli
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