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Search Results for " ace inhibitor "
Targets Recommended: RAAS

101

抑制剂 & 化合物

11

天然产物

1

重组蛋白

8

同位素标记化合物

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Cat. No. Product Name Target Signaling Pathways
T7686 Ramiprilat

RAAS Endocrinology/Hormones
Ramiprilat 是 Ramipril 的活性代谢物,是一种口服有活力的血管紧张素转换酶 (ACE) 抑制剂,其 Ki=7 pM。它可用于研究心力衰竭以及高血压。
T7510 Leucylarginylproline

RAAS Endocrinology/Hormones
Leucylarginylproline 是一种血管紧张素转换酶抑制剂,IC50=为0.27μM。
T1484 Perindoprilat

Perindoprilate,培哚普利

RAAS; MRP; AChR Endocrinology/Hormones; Immunology/Inflammation; Neuroscience
Perindoprilat (Perindoprilate) 是一种血管紧张素转换酶抑制剂。
T1605 Enalapril

MK-421,依那普利

RAAS; MRP Endocrinology/Hormones; Immunology/Inflammation
Enalapril 是一种血管紧张素转换酶(ACE)抑制剂。
T13865 Resorcinolnaphthalein

RAAS Endocrinology/Hormones
Resorcinolnaphthalein 是一种特异性的血管紧张素转换酶 2 激活剂,EC50=19.5 μM。Resorcinolnaphthalein 能够用于高血压和肾纤维化的研究
T16116 MLN-4760

RAAS Endocrinology/Hormones
MLN-4760 是选择性的人ACE2抑制剂,IC50=0.44 nM,对人ACE2的选择性是其他相关蛋白的 5000 多倍,包括人睾丸 ACE (IC50,>100 μM) 和牛 carboxypeptidase A (IC50,27 μM)。
T1145 Diminazene Aceturate

DIZE

Others; Serine Protease; Parasite Microbiology/Virology; Others; Proteases/Proteasome
Diminazene aceturate 是血管紧张素转化酶 2 的激活剂,具有强效抗炎特性。它还是一种抗锥虫药物,适用于牲畜。它主要生化机理是通过与富含腺嘌呤-胸腺嘧啶碱基对的位点发生特异性相互作用,以非插入方式与锥虫动子体 DNA 结合。
T1489 Fosinopril sodium

SQ28555,福辛普利钠

RAAS Endocrinology/Hormones
Fosinopril sodium 是一种血管紧张素转换酶(ACE)抑制剂的前药,能够作用于高血压和慢性心力衰竭。
TP1828 N-Acetyl-Ser-Asp-Lys-Pro

RAAS Endocrinology/Hormones
N-Acetyl-Ser-Asp-Lys-Pro 通过酶促处理胸腺素 β4 在骨髓细胞中形成。 它抑制多能造血干细胞进入细胞周期的 S 期,并防止小鼠中的 Ara-C 致死性。
T3281 Delapril hydrochloride

indalapril,地拉普利盐酸盐,Alindapril Hydrochloride,Delapril Hydrochloride,盐酸地拉普利,CV 3317

RAAS Endocrinology/Hormones
Delapril hydrochloride (indalapril) 是一种血管紧张素转化酶抑制剂,能够用于心血管疾病的研究。
T7808 Alacepril

Cetapril,阿拉普利,DU-1219

RAAS Endocrinology/Hormones
Alacepril (DU-1219) 是一种具有口服活性血管紧张素转换酶 (ACE) 抑制剂,具有长效抗高血压作用。
T1645 Ramipril

HOE-498,Tritace,雷米普利,Altace,Carasel

Apoptosis; RAAS Apoptosis; Endocrinology/Hormones
Ramipril (Altace) 是一种ACE 抑制剂,IC50为5 nM。
T5030 Zofenopril calcium

SQ26991,佐芬普利钙,Zofenopril (calcium)

RAAS; Reactive Oxygen Species Endocrinology/Hormones; Immunology/Inflammation; Metabolism; NF-κB
Zofenopril calcium (SQ26991) 是一种抗氧化剂和血管紧张素转化酶 (ACE) 抑制剂。
T2486 IOWH-032

IOWH032,IOWH 032

CFTR; Autophagy Autophagy; Membrane transporter/Ion channel
IOWH-032 (IOWH032) 是一种合成 CFTR 抑制剂,可用于研究治疗霍乱、腹泻和分泌性腹泻,在T84和CHO-CFTR 细胞实验中IC50为1.01 uM。
T0180 Benazepril hydrochloride

盐酸贝那普利,CGS 14824A HCl,Benazepril HCl,CGS14824A

RAAS Endocrinology/Hormones
Benazepril hydrochloride (CGS 14824A HCl) 是一种血管紧张素转化酶(ACE)抑制剂,能够作用于高血压。
T2679 BMS-265246

BMS265246

CDK Cell Cycle/Checkpoint
BMS-265246 是一种有效的选择性 CDK1/2 抑制剂,对 CDK1/cyclin B 和 CDK2/cyclin E 的 IC50分别为6 nM 和9 nM。
T5329 Trandolapril

Angiotensin-converting Enzyme (ACE) Metabolism
Trandolapril 是 Trandolaprilat 的前体药物。Trandolapril 是一种口服血管紧张素转换酶抑制剂,在高血压和充血性心力衰竭及心肌梗死领域有研究价值。
T0706 Lisinopril dihydrate

Lisinopril,Renacor,赖诺普利二水合物,MK-521 (dihydrate)

RAAS; MRP Endocrinology/Hormones; Immunology/Inflammation
Lisinopril dihydrate (MK-521) 是一种血管紧张素转化酶抑制剂。Lisinopri dihydrate 能够作用于高血压,充血性心力衰竭和心脏病等。
T7714 Temocapil

Tyrosinase Proteases/Proteasome
Temocapil 是一种酪氨酸激酶抑制剂。
T0805 Quinapril hydrochloride

CI-906,PD-109452-2,盐酸喹那普利,Quinapril HCl

RAAS Endocrinology/Hormones
Quinapril hydrochloride (PD-109452-2) 是一种血管紧张素转化酶(ACE) 抑制剂的原药。
T6542 Imidapril hydrochloride

Novaloc,Imidapril HCl,盐酸咪达普利,Tanapril,TA-6366

RAAS Endocrinology/Hormones
Imidapril hydrochloride (Tanapril) 是一种血管紧张素转换酶 (ACE) 抑制剂,具有抗高血压活性。
T6340 Enalaprilat Dihydrate

依那普利拉二水合物,MK-422,MK-422 Dihydrate

RAAS; Autophagy Autophagy; Endocrinology/Hormones
Enalaprilat Dihydrate (MK-422 Dihydrate) 是一种有效的血管紧张素转化酶抑制剂,IC50为 1.94 nM。
T1462 Captopril

SQ 14225,甲巯丙脯酸,卡托普利,SQ-14534,SA333

RAAS Endocrinology/Hormones
Captopril (SA333) 是一种含巯基的,具有口服活性的血管紧张素转换酶(ACE)抑制剂 ,IC50=0.025 μM,广泛应用于高血压和充血性心力衰竭的研究。Captopril 也是NDM-1抑制剂,IC50=7.9 μM。
T1484L Perindopril erbumine

培哚普利叔丁胺,培哚普利叔丁胺盐,S9490-3,Perindopril tert-butylamine salt

Apoptosis; RAAS; MRP Apoptosis; Endocrinology/Hormones; Immunology/Inflammation
Perindopril erbumine (S9490-3) 是一种长效血管紧张素转换酶抑制剂。
T7339 Angiotensin (1-7)

Ang-(1-7),Angiotensin 1-7,ASP-ARG-VAL-TYR-ILE-HIS-PRO

RAAS; Endogenous Metabolite Endocrinology/Hormones; Metabolism
Angiotensin (1-7) (ASP-ARG-VAL-TYR-ILE-HIS-PRO) 是肾素-血管紧张素系统中的内源性七肽。Angiotensin 1-7在心肌细胞中具有抗炎和抗纤维化活性,因此具有心脏保护作用。它能抑制血管紧张素转换酶和释放一氧化氮,是激肽诱导的血管舒张的局部协同调节剂。它阻断 Ang II 诱导的平滑肌细胞增殖和肥大,并显示对内皮的抗血管生成和生长抑制作用。它显示出抗炎活性。
T6486 Enalapril Maleate

MK-421 Maleate,Renitec Maleate,Glioten Maleate,MK-421 (maleate),Vasotec Maleate,马来酸依那普利

RAAS Endocrinology/Hormones
Enalapril Maleate (MK-421 Maleate) 一种是血管紧张素转化酶(ACE)抑制剂。
T6595 Moexipril hydrochloride

莫昔普利盐酸盐,Moexipril HCl,RS-10085,SPM 925,CI-925

Apoptosis; RAAS Apoptosis; Endocrinology/Hormones
Moexipril hydrochloride (Moexipril HCl) 是一种有口服活性的,不含巯基的血管紧张素转化酶抑制剂,可治疗高血压和充血性心力衰竭。
T6698 Temocapril hydrochloride

CS-622 HCl,Acecol,Temocapril HCl,CS-622,盐酸替莫普利

RAAS Endocrinology/Hormones
Temocapril hydrochloride (CS-622 HCl) 是血管紧张素转化酶 (ACE) 抑制剂。Temocapril HCl 能够用于充血性心力衰竭、急性心肌梗死、高血压、胰岛素抵抗和肾脏疾病的研究。
T6444 Cilazapril Monohydrate

Ro 31-2848 monohydrate,Justor,西拉普利,西拉普利水合物

RAAS Endocrinology/Hormones
Cilazapril Monohydrate (Justor) 是一种血管紧张素转化酶抑制剂,能够作用于高血压和充血性心力衰竭的研究。
TP1622 DX600 TFA

RAAS Endocrinology/Hormones
DX600 TFA 是 ACE2 的特异性抑制剂,不会与 ACE 发生交叉反应。
T20689 Temocaprilat

RNH-5139,RS-5139,RNH 5139,RNH5139,替莫普利,RS5139,RS 5139

Angiotensin-converting Enzyme (ACE) Metabolism
Temocaprilat (RS5139) 是一种血管紧张素转换酶 (ACE) 抑制剂。 Temocaprilat 通过缺乏 EHBR 的 cMOAT 有效地从胆汁中排泄,而许多其他 ACE 抑制剂对 cMOAT 的亲和力较低。
T7354 H-Val-Pro-Pro-OH

RAAS Endocrinology/Hormones
H-Val-Pro-Pro-OH 是一种血管紧张素 I 转化酶(ACE)的抑制剂(IC50:9 μM)。他是一种来源于牛奶的脯氨酸肽衍生物。
T24906L Tuna AI acetate

Angiotensin-converting Enzyme (ACE) Metabolism
Tuna AI acetate 是一种源自金枪鱼肌肉的非竞争性血管紧张素转换酶 (ACE) 抑制剂。
TP1750L H-Ile-Pro-Pro-OH acetate

H-Ile-Pro-Pro-OH acetate(26001-32-1 free base)

Angiotensin-converting Enzyme (ACE) Metabolism
H-Ile-Pro-Pro-OH acetate 是一种血管紧张素转换酶抑制剂,为乳源三肽。
T25226 Ceronapril

Ceronaprilum,SQ 29852,SQ-29852,SQ29852

RAAS Endocrinology/Hormones
Ceronapril (SQ 29852) 是一种具有口服活性和高效性的血管紧张素转换酶 (ACE) 抑制剂(IC50 : 36 nM),可用于研究痴呆和高血压。
T11175 Elenbecestat

E2609

Beta-Secretase; BACE Neuroscience
Elenbecestat (E2609) 是一种高效、有口服活性的,能透过 CNS 的 BACE-1抑制剂,它有用于阿尔茨海默病 (AD) 的研究潜力。
T26213 SQ 27786

SQ27,786,SQ27786,SQ-27786,SQ-27,786,SQ 27,786

Others Others
SQ 27786 is an inhibitor of ACE.
T26067 Rev 6207

Rev-6207

Others Others
Rev 6207 is a non-sulfhydryl ACE-inhibitor.
T25178 Brl 36378

Brl36378,Brl-36378

Others Others
Brl 36378 is an inhibitor of ACE.
T26065 Rev 5975

Others Others
Rev 5975 is a non-sulfhydryl ACE-inhibitor.
T27608 Indolapril hydrochloride

REV 6000A(SS),CI-907,CI 907,CI907,Indolapril HCl

Others Others
Indolapril hydrochloride is a nonsulfhydryl angiotensin converting enzyme (ACE) inhibitor with antihypertensive activity.
T13274 Utibapril

FPL 63547

Others Others
Utibapril is an inhibitor of angiotensin-converting enzyme (ACE) with antihypertensive activities.
T71028 Lisinopril, epsilon-biotinamidocaproyl-

Others Others
Lisinopril, epsilon-biotinamidocaproyl- is an angiotensin converting enzyme (ACE) inhibitor.
T25801 Methylsilanol acetyltyrosine

Tyrosilane

Others Others
Methylsilanol acetyltyrosine is used as an ACE inhibitor.
T70698 MDL-100173

Others Others
MDL-100173 is a dual angiotensin-converting enzyme (ACE)/neutral endopeptidase (NEP) inhibitor.
T68435 Cilazapril HCl

Others Others
Cilazapril, also known as Ro 31 2848, is a potent ACE inhibitor used for hypertension. Cilazapril is a prodrug that is hydrolyzed after absorption to its main metabolite cilazaprilat. Cilazapril is a monoethyl ester, which acts as an angiotensin-converting enzyme (ACE) inhibitor. The inhibitor functions by inhibiting the ability of ACE to cleave bonds of angiotensin I and Hip-His-Leu. It is known that the diacid form of Cilazapril is more potent that enalapril at inhibiting ACE.
T28037 Microginin 527

Others Others
Microginin 527, a compound found in Microcystis, is an inhibitor of protein phosphatase, ACE, and leucine aminopeptidase.
T25564 K-13

K-13 (Ace inhib)

Others Others
K-13 is used as an ACE inhibitor produced by Micromonospora halophytics subsp. exilisia K-13.
T25449 GF 109

GF109,GF-109

Others Others
GF 109 is an inhibitor of ACE.
T68533 Moveltipril calcium salt

Others Others
Moveltipril calcium salt is an ACE inhibitor.

化合物

Ramiprilat
Cat.No: T7686
Synonym:
Target: RAAS
Leucylarginylproline
Cat.No: T7510
Synonym:
Target: RAAS
Perindoprilat
Cat.No: T1484
Synonym: Perindoprilate,培哚普利
Target: RAAS, MRP, AChR
Enalapril
Cat.No: T1605
Synonym: MK-421,依那普利
Target: RAAS, MRP
Resorcinolnaphthalein
Cat.No: T13865
Synonym:
Target: RAAS
MLN-4760
Cat.No: T16116
Synonym:
Target: RAAS
Diminazene Aceturate
Cat.No: T1145
Synonym: DIZE
Target: Others, Serine Protease, Parasite
Fosinopril sodium
Cat.No: T1489
Synonym: SQ28555,福辛普利钠
Target: RAAS
N-Acetyl-Ser-Asp-Lys-Pro
Cat.No: TP1828
Synonym:
Target: RAAS
Delapril hydrochloride
Cat.No: T3281
Synonym: indalapril,地拉普利盐酸盐,Alindapril Hydrochloride,Delapril Hydrochloride,盐酸地拉普利,CV 3317
Target: RAAS
Alacepril
Cat.No: T7808
Synonym: Cetapril,阿拉普利,DU-1219
Target: RAAS
Ramipril
Cat.No: T1645
Synonym: HOE-498,Tritace,雷米普利,Altace,Carasel
Target: Apoptosis, RAAS
Zofenopril calcium
Cat.No: T5030
Synonym: SQ26991,佐芬普利钙,Zofenopril (calcium)
Target: RAAS, Reactive Oxygen Species
IOWH-032
Cat.No: T2486
Synonym: IOWH032,IOWH 032
Target: CFTR, Autophagy
Benazepril hydrochloride
Cat.No: T0180
Synonym: 盐酸贝那普利,CGS 14824A HCl,Benazepril HCl,CGS14824A
Target: RAAS
BMS-265246
Cat.No: T2679
Synonym: BMS265246
Target: CDK
Trandolapril
Cat.No: T5329
Synonym:
Target: Angiotensin-converting Enzyme (ACE)
Lisinopril dihydrate
Cat.No: T0706
Synonym: Lisinopril,Renacor,赖诺普利二水合物,MK-521 (dihydrate)
Target: RAAS, MRP
Temocapil
Cat.No: T7714
Synonym:
Target: Tyrosinase
Quinapril hydrochloride
Cat.No: T0805
Synonym: CI-906,PD-109452-2,盐酸喹那普利,Quinapril HCl
Target: RAAS
Imidapril hydrochloride
Cat.No: T6542
Synonym: Novaloc,Imidapril HCl,盐酸咪达普利,Tanapril,TA-6366
Target: RAAS
Enalaprilat Dihydrate
Cat.No: T6340
Synonym: 依那普利拉二水合物,MK-422,MK-422 Dihydrate
Target: RAAS, Autophagy
Captopril
Cat.No: T1462
Synonym: SQ 14225,甲巯丙脯酸,卡托普利,SQ-14534,SA333
Target: RAAS
Perindopril erbumine
Cat.No: T1484L
Synonym: 培哚普利叔丁胺,培哚普利叔丁胺盐,S9490-3,Perindopril tert-butylamine salt
Target: Apoptosis, RAAS, MRP
Angiotensin (1-7)
Cat.No: T7339
Synonym: Ang-(1-7),Angiotensin 1-7,ASP-ARG-VAL-TYR-ILE-HIS-PRO
Target: RAAS, Endogenous Metabolite
Enalapril Maleate
Cat.No: T6486
Synonym: MK-421 Maleate,Renitec Maleate,Glioten Maleate,MK-421 (maleate),Vasotec Maleate,马来酸依那普利
Target: RAAS
Moexipril hydrochloride
Cat.No: T6595
Synonym: 莫昔普利盐酸盐,Moexipril HCl,RS-10085,SPM 925,CI-925
Target: Apoptosis, RAAS
Temocapril hydrochloride
Cat.No: T6698
Synonym: CS-622 HCl,Acecol,Temocapril HCl,CS-622,盐酸替莫普利
Target: RAAS
Cilazapril Monohydrate
Cat.No: T6444
Synonym: Ro 31-2848 monohydrate,Justor,西拉普利,西拉普利水合物
Target: RAAS
DX600 TFA
Cat.No: TP1622
Synonym:
Target: RAAS
Temocaprilat
Cat.No: T20689
Synonym: RNH-5139,RS-5139,RNH 5139,RNH5139,替莫普利,RS5139,RS 5139
Target: Angiotensin-converting Enzyme (ACE)
H-Val-Pro-Pro-OH
Cat.No: T7354
Synonym:
Target: RAAS
Tuna AI acetate
Cat.No: T24906L
Synonym:
Target: Angiotensin-converting Enzyme (ACE)
H-Ile-Pro-Pro-OH acetate
Cat.No: TP1750L
Synonym: H-Ile-Pro-Pro-OH acetate(26001-32-1 free base)
Target: Angiotensin-converting Enzyme (ACE)
Ceronapril
Cat.No: T25226
Synonym: Ceronaprilum,SQ 29852,SQ-29852,SQ29852
Target: RAAS
Elenbecestat
Cat.No: T11175
Synonym: E2609
Target: Beta-Secretase, BACE
SQ 27786
Cat.No: T26213
Synonym: SQ27,786,SQ27786,SQ-27786,SQ-27,786,SQ 27,786
Target: Others
Rev 6207
Cat.No: T26067
Synonym: Rev-6207
Target: Others
Brl 36378
Cat.No: T25178
Synonym: Brl36378,Brl-36378
Target: Others
Rev 5975
Cat.No: T26065
Synonym:
Target: Others
Indolapril hydrochloride
Cat.No: T27608
Synonym: REV 6000A(SS),CI-907,CI 907,CI907,Indolapril HCl
Target: Others
Utibapril
Cat.No: T13274
Synonym: FPL 63547
Target: Others
Lisinopril, epsilon-biotinamidocaproyl-
Cat.No: T71028
Synonym:
Target: Others
Methylsilanol acetyltyrosine
Cat.No: T25801
Synonym: Tyrosilane
Target: Others
MDL-100173
Cat.No: T70698
Synonym:
Target: Others
Cilazapril HCl
Cat.No: T68435
Synonym:
Target: Others
Microginin 527
Cat.No: T28037
Synonym:
Target: Others
K-13
Cat.No: T25564
Synonym: K-13 (Ace inhib)
Target: Others
GF 109
Cat.No: T25449
Synonym: GF109,GF-109
Target: Others
Moveltipril calcium salt
Cat.No: T68533
Synonym:
Target: Others
Cat. No. Product Name Target Signaling Pathways
T13299 Vicenin 3

维采宁-3,维采宁 3

RAAS Endocrinology/Hormones
Vicenin 3来源于广金钱草的地上部分。Vicenin 3是血管紧张素转换酶抑制剂,IC50=46.91 μM。
T8270 Deserpidine

地舍平,Harmonyl

RAAS Endocrinology/Hormones
Deserpidine (Harmonyl) 是从 Rauwolfia canescens 的根中分离的生物碱。Deserpidine 与 Reserpine 相关。Deserpidine 是竞争性血管紧张素转化酶抑制剂,可以被用作抗高血压药以及镇定剂。Deserpidine 还减少了肾上腺皮质血管紧张素 II 诱导的醛固酮分泌。
T5S0106 Peimisine

贝母辛,Ebeiensine

RAAS; AChR Endocrinology/Hormones; Neuroscience
Peimisine (Ebeiensine) 非竞争性拮抗气管平滑肌 M 受体,抑制 Ach 引起的平滑肌收缩。它兴奋 β 受体和拮抗内钙释放,促进一氧化氮释放,可舒张气管平滑肌,有平喘作用。
T5796 Plantainoside D

Isoplantamajoside,车前草苷D

RAAS; PKC Chromatin/Epigenetic; Cytoskeletal Signaling; Endocrinology/Hormones
Plantainoside D (Isoplantamajoside) 可以抑制 ACE ,IC50=2.17 mM。Plantainoside D 也是IKK-β抑制剂。
T21418 Lisinopril

Linopril,赖诺普利,Zestril,Prinivil,Lisipril

RAAS Endocrinology/Hormones
Lisinopril (Prinivil) 是一种血管紧张素转化酶抑制剂,能够作用于高血压,充血性心力衰竭和心脏病等。
T3851 Vicenin 2

Vicenin -2,维采宁 2,新西兰牡荆苷

RAAS Endocrinology/Hormones
Vicenin 2 来源于广金钱草 (Desmodium styracifolium) 的地上部分。Vicenin 2 是一种血管紧张素转换酶 (ACE) 抑制剂,IC50=43.83 μM。
T3753 Sinapinic Acid

Sinapic acid,芥子酸,Synapoic acid

Apoptosis; RAAS; Reactive Oxygen Species; HDAC Apoptosis; Chromatin/Epigenetic; DNA Damage/DNA Repair; Endocrinology/Hormones; Immunology/Inflammation; Metabolism; NF-κB
Sinapinic Acid (Synapoic acid) 是从 Hydnophytum formicarumJack. 根中分离到的酚类,是HDAC 抑制剂,对ACE-I 的活性也有抑制作用。它有抗肿瘤活性,诱导肿瘤细胞凋亡,具有抗氧化、抗糖尿病的作用。
T6627 Phosphoramidon Disodium

Phosphoramidon Disodium Salt,磷酰胺二钠

RAAS; Neprilysin; Others Endocrinology/Hormones; Metabolism; Others
Phosphoramidon Disodium (Phosphoramidon Disodium Salt) Salt 是一种金属蛋白酶 (metalloprotease) 抑制剂 。Phosphoramidon Disodium Salt 抑制内皮素转化酶 (ECE) ,中性肽内切酶 (NEP) 和血管紧张素转换酶 (ACE) 的IC50分别为 3.5 ,0.034 和 78 μM。
T38481 Camellianin B

Others Others
Camellianin B, a flavonoid compound and metabolite of Camellianin A, exhibits antioxidant properties and acts as an angiotensin converting enzyme (ACE) inhibitor.
T79958 Isocrenatoside

Angiotensin-converting Enzyme (ACE) Metabolism
Isocrenatoside (compound 6)为环状八肽,具有ACE抑制活性。该化合物可通过乙醇提取Microtoena prainiana茎部分离纯化。研究显示,1 mg/mL浓度下,Isocrenatoside的ACE抑制效率高达99.3%。
TN1104 Cyanidin 3-sambubioside chloride

Cyanidin-3-O-sambubioside chloride

RAAS; Antioxidant; NO Synthase Endocrinology/Hormones; Immunology/Inflammation; oxidation-reduction
Cyanidin 3-sambubioside chloride (Cyanidin-3-O-sambubioside chloride) 是一种从植物中提取的花青素,是一种 NO和 H274Y 突变的抑制剂,对流感神经氨酸酶具有抑制作用。Cyanidin 3-sambubioside chloride 具有抗氧化,抗血管生成和抗病毒活性,抑制血管紧张素转换酶 (ACE) 的活性,可用于研究病毒感染和心血管疾病。

天然产物

Vicenin 3
Cat.No: T13299
Synonym: 维采宁-3,维采宁 3
Target: RAAS
Deserpidine
Cat.No: T8270
Synonym: 地舍平,Harmonyl
Target: RAAS
Peimisine
Cat.No: T5S0106
Synonym: 贝母辛,Ebeiensine
Target: RAAS, AChR
Plantainoside D
Cat.No: T5796
Synonym: Isoplantamajoside,车前草苷D
Target: RAAS, PKC
Lisinopril
Cat.No: T21418
Synonym: Linopril,赖诺普利,Zestril,Prinivil,Lisipril
Target: RAAS
Vicenin 2
Cat.No: T3851
Synonym: Vicenin -2,维采宁 2,新西兰牡荆苷
Target: RAAS
Sinapinic Acid
Cat.No: T3753
Synonym: Sinapic acid,芥子酸,Synapoic acid
Target: Apoptosis, RAAS, Reactive Oxygen Species, HDAC
Phosphoramidon Disodium
Cat.No: T6627
Synonym: Phosphoramidon Disodium Salt,磷酰胺二钠
Target: RAAS, Neprilysin, Others
Camellianin B
Cat.No: T38481
Synonym:
Target: Others
Isocrenatoside
Cat.No: T79958
Synonym:
Target: Angiotensin-converting Enzyme (ACE)
Cyanidin 3-sambubioside chloride
Cat.No: TN1104
Synonym: Cyanidin-3-O-sambubioside chloride
Target: RAAS, Antioxidant, NO Synthase
Cat. No. Product Name Species Expression System
TMPJ-00386 ACE2/ACEH Protein, Human, Recombinant (HEK293, His & Avi), Biotinylated

Metalloprotease MPROT15,ACEH,Angiotensin-Converting...

Human HEK293 Cells
Angiotensin-Converting Enzyme 2 (ACE-2) is an integral membrane protein and a zinc metalloprotease of the ACE family, the ACE family includes somatic and germinal ACE. ACE-2 cleaves angiotensins I and II as a carboxypeptidase, ACE-2 converts angiotensin I to angiotensin 1-9, and angiotensin II to angiotensin 1-7. ACE-2 is also able to hydrolyze apelin-13 and dynorphin-13 with high efficiency. ACE-2 can be high expressed in testis, kidney and heart, in colon, small intestine and ovary at moderate...

重组蛋白

ACE2/ACEH Protein, Human, Recombinant (HEK293, His & Avi), Biotinylated
Cat.No: TMPJ-00386
Species: Human
Expression System: HEK293 Cells
Cat. No. Product Name Target Signaling Pathways
T11192 Enalapril D5 maleate

MK-421 D5 maleate,马来酸依那普利D5

Others Others
Enalapril D5 maleate is deuterium labeled Enalapril, which is an angiotensin converting enzyme (ACE) inhibitor.
T11194 Enalaprilat D5

MK-422 D5,依那普利拉 D5

Others Others
Enalaprilat D5 is the deuterium labeled Enalaprilat, which is an angiotensin-converting enzyme (ACE) inhibitor.
T11193 Enalaprilat-d5 sodium

MK-422 D5 Sodium Salt,依那普利拉钠 D5,Enalaprilat D5 Sodium Salt

Others Others
Enalaprilat D5 Sodium Salt is the deuterium labeled Enalaprilat, which is an angiotensin-converting enzyme (ACE) inhibitor.
T13196 Trandolaprilate D5

Trandolaprilat D5,RU 44403 D5

Others Others
Trandolaprilate D5 is a deuterium-labeled Trandolaprilate. Trandolaprilate is an inhibitor of angiotensin-converting enzyme (ACE).
T13195 Trandolapril D5

RU44570 D5

Others Others
Trandolapril D5 is a deuterium labeled Trandolapril. Trandolapril is an orally active inhibitor of angiotensin converting enzyme (ACE) for hypertension and congestive heart failure (CHF).
TMIJ-0253 Benazepril-d5 HCl

Benazepril-d5 HCl 是 Benazepril HCl 的氘代化合物。Benazepril HCl 的 CAS 号为 86541-74-4。Benazepril hydrochloride 是一种血管紧张素转化酶(ACE)抑制剂,能够作用于高血压。
T70883 Moexipril-d5

Moexipril-d5 intended for use as an internal standard for the quantification of moexipril by GC- or LC-MS. Moexipril is a prodrug form of the angiotensin converting enzyme (ACE) inhibitor moexiprilat. It is converted to moexiprilat in vivo by side chain ester hydrolysis. Moexipril inhibits ACE in a cell-free assay (IC50 = 2.7 µM for the rabbit enzyme). It also inhibits phosphodiesterase 4 (IC50s = 38, 160, and 230 µM for PDE4B2, PDE4A5 and PDE4D5, respectively). Moexipril (0.1-30 mg/kg per day) ...
T71065 Quinapril-d5

Quinapril-d5 is intended for use as an internal standard for the quantification of quinapril by GC- or LC-MS. Quinapril is a prodrug form of the angiotensin converting enzyme (ACE) inhibitor quinaprilat. In vivo, quinapril reduces mean arterial pressure in renal hypertensive and spontaneously hypertensive rats. It inhibits angiotensin I-induced pressor responses in normotensive rats and dogs. Quinapril prevents left ventricular heart failure in CHF 14.6 cardiomyopathic hamsters. Formulations con...

同位素标记化合物

Enalapril D5 maleate
Cat.No: T11192
Synonym: MK-421 D5 maleate,马来酸依那普利D5
Target: Others
Enalaprilat D5
Cat.No: T11194
Synonym: MK-422 D5,依那普利拉 D5
Target: Others
Enalaprilat-d5 sodium
Cat.No: T11193
Synonym: MK-422 D5 Sodium Salt,依那普利拉钠 D5,Enalaprilat D5 Sodium Salt
Target: Others
Trandolaprilate D5
Cat.No: T13196
Synonym: Trandolaprilat D5,RU 44403 D5
Target: Others
Trandolapril D5
Cat.No: T13195
Synonym: RU44570 D5
Target: Others
Benazepril-d5 HCl
Cat.No: TMIJ-0253
Synonym:
Target:
Moexipril-d5
Cat.No: T70883
Synonym:
Target:
Quinapril-d5
Cat.No: T71065
Synonym:
Target:
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