2646
709
1
51
61
Cat. No. | Product Name | Form | Specificity Of Inhibition |
---|---|---|---|
C0048 |
Deacetylase Inhibitor Cocktail (100× in 70% DMSO)
去乙酰化酶抑制剂 Cocktail(100× in 70% DMSO) |
Solution (100× in 70% DMSO) | Class I/II/III HDAC |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T77457 |
Emicizumab
ACE 910,RO 5534262 |
Others | Others |
Emicizumab(ACE 910) 是一种人源化单克隆抗体,桥接活化因子 IX 和激活因子 X,以模拟活化因子 VIII 的功能。Emicizumab 可用于预防和治疗血友病 A 。 | |||
T32366 |
Kaya-ace
NK 0795,BRN 2169649 |
Others | Others |
Kaya-ace is a bioactive chemical. | |||
T25564 |
K-13
K-13 (Ace inhib) |
Others | Others |
K-13 is used as an ACE inhibitor produced by Micromonospora halophytics subsp. exilisia K-13. | |||
T7686 |
Ramiprilat
|
RAAS | Endocrinology/Hormones |
Ramiprilat 是 Ramipril 的活性代谢物,是一种口服有活力的血管紧张素转换酶 (ACE) 抑制剂,其 Ki=7 pM。它可用于研究心力衰竭以及高血压。 | |||
T7510 |
Leucylarginylproline
|
RAAS | Endocrinology/Hormones |
Leucylarginylproline 是一种血管紧张素转换酶抑制剂,IC50=为0.27μM。 | |||
T1484 |
Perindoprilat
Perindoprilate,培哚普利 |
RAAS; MRP; AChR | Endocrinology/Hormones; Immunology/Inflammation; Neuroscience |
Perindoprilat (Perindoprilate) 是一种血管紧张素转换酶抑制剂。 | |||
T1605 |
Enalapril
MK-421,依那普利 |
RAAS; MRP | Endocrinology/Hormones; Immunology/Inflammation |
Enalapril 是一种血管紧张素转换酶(ACE)抑制剂。 | |||
T13865 |
Resorcinolnaphthalein
|
RAAS | Endocrinology/Hormones |
Resorcinolnaphthalein 是一种特异性的血管紧张素转换酶 2 激活剂,EC50=19.5 μM。Resorcinolnaphthalein 能够用于高血压和肾纤维化的研究 | |||
T1489 |
Fosinopril sodium
SQ28555,福辛普利钠 |
RAAS | Endocrinology/Hormones |
Fosinopril sodium 是一种血管紧张素转换酶(ACE)抑制剂的前药,能够作用于高血压和慢性心力衰竭。 | |||
T1145 |
Diminazene Aceturate
DIZE |
Others; Serine Protease; Parasite | Microbiology/Virology; Others; Proteases/Proteasome |
Diminazene aceturate 是血管紧张素转化酶 2 的激活剂,具有强效抗炎特性。它还是一种抗锥虫药物,适用于牲畜。它主要生化机理是通过与富含腺嘌呤-胸腺嘧啶碱基对的位点发生特异性相互作用,以非插入方式与锥虫动子体 DNA 结合。 | |||
T16116 |
MLN-4760
|
RAAS | Endocrinology/Hormones |
MLN-4760 是选择性的人ACE2抑制剂,IC50=0.44 nM,对人ACE2的选择性是其他相关蛋白的 5000 多倍,包括人睾丸 ACE (IC50,>100 μM) 和牛 carboxypeptidase A (IC50,27 μM)。 | |||
TP1828 |
N-Acetyl-Ser-Asp-Lys-Pro
|
RAAS | Endocrinology/Hormones |
N-Acetyl-Ser-Asp-Lys-Pro 通过酶促处理胸腺素 β4 在骨髓细胞中形成。 它抑制多能造血干细胞进入细胞周期的 S 期,并防止小鼠中的 Ara-C 致死性。 | |||
T3281 |
Delapril hydrochloride
indalapril,地拉普利盐酸盐,Alindapril Hydrochloride,Delapril Hydrochloride,盐酸地拉普利,CV 3317 |
RAAS | Endocrinology/Hormones |
Delapril hydrochloride (indalapril) 是一种血管紧张素转化酶抑制剂,能够用于心血管疾病的研究。 | |||
T7808 |
Alacepril
Cetapril,阿拉普利,DU-1219 |
RAAS | Endocrinology/Hormones |
Alacepril (DU-1219) 是一种具有口服活性血管紧张素转换酶 (ACE) 抑制剂,具有长效抗高血压作用。 | |||
T1645 |
Ramipril
HOE-498,Tritace,雷米普利,Altace,Carasel |
Apoptosis; RAAS | Apoptosis; Endocrinology/Hormones |
Ramipril (Altace) 是一种ACE 抑制剂,IC50为5 nM。 | |||
T5030 |
Zofenopril calcium
SQ26991,佐芬普利钙,Zofenopril (calcium) |
RAAS; Reactive Oxygen Species | Endocrinology/Hormones; Immunology/Inflammation; Metabolism; NF-κB |
Zofenopril calcium (SQ26991) 是一种抗氧化剂和血管紧张素转化酶 (ACE) 抑制剂。 | |||
T0180 |
Benazepril hydrochloride
盐酸贝那普利,CGS 14824A HCl,Benazepril HCl,CGS14824A |
RAAS | Endocrinology/Hormones |
Benazepril hydrochloride (CGS 14824A HCl) 是一种血管紧张素转化酶(ACE)抑制剂,能够作用于高血压。 | |||
T2486 |
IOWH-032
IOWH032,IOWH 032 |
CFTR; Autophagy | Autophagy; Membrane transporter/Ion channel |
IOWH-032 (IOWH032) 是一种合成 CFTR 抑制剂,可用于研究治疗霍乱、腹泻和分泌性腹泻,在T84和CHO-CFTR 细胞实验中IC50为1.01 uM。 | |||
T2679 |
BMS-265246
BMS265246 |
CDK | Cell Cycle/Checkpoint |
BMS-265246 是一种有效的选择性 CDK1/2 抑制剂,对 CDK1/cyclin B 和 CDK2/cyclin E 的 IC50分别为6 nM 和9 nM。 | |||
T5329 |
Trandolapril
|
Angiotensin-converting Enzyme (ACE) | Metabolism |
Trandolapril 是 Trandolaprilat 的前体药物。Trandolapril 是一种口服血管紧张素转换酶抑制剂,在高血压和充血性心力衰竭及心肌梗死领域有研究价值。 | |||
T0706 |
Lisinopril dihydrate
Lisinopril,Renacor,赖诺普利二水合物,MK-521 (dihydrate) |
RAAS; MRP | Endocrinology/Hormones; Immunology/Inflammation |
Lisinopril dihydrate (MK-521) 是一种血管紧张素转化酶抑制剂。Lisinopri dihydrate 能够作用于高血压,充血性心力衰竭和心脏病等。 | |||
T7714 |
Temocapil
|
Tyrosinase | Proteases/Proteasome |
Temocapil 是一种酪氨酸激酶抑制剂。 | |||
T0805 |
Quinapril hydrochloride
CI-906,PD-109452-2,盐酸喹那普利,Quinapril HCl |
RAAS | Endocrinology/Hormones |
Quinapril hydrochloride (PD-109452-2) 是一种血管紧张素转化酶(ACE) 抑制剂的原药。 | |||
T6542 |
Imidapril hydrochloride
Novaloc,Imidapril HCl,盐酸咪达普利,Tanapril,TA-6366 |
RAAS | Endocrinology/Hormones |
Imidapril hydrochloride (Tanapril) 是一种血管紧张素转换酶 (ACE) 抑制剂,具有抗高血压活性。 | |||
T6340 |
Enalaprilat Dihydrate
依那普利拉二水合物,MK-422,MK-422 Dihydrate |
RAAS; Autophagy | Autophagy; Endocrinology/Hormones |
Enalaprilat Dihydrate (MK-422 Dihydrate) 是一种有效的血管紧张素转化酶抑制剂,IC50为 1.94 nM。 | |||
T1462 |
Captopril
SQ 14225,甲巯丙脯酸,卡托普利,SQ-14534,SA333 |
RAAS | Endocrinology/Hormones |
Captopril (SA333) 是一种含巯基的,具有口服活性的血管紧张素转换酶(ACE)抑制剂 ,IC50=0.025 μM,广泛应用于高血压和充血性心力衰竭的研究。Captopril 也是NDM-1抑制剂,IC50=7.9 μM。 | |||
T1484L |
Perindopril erbumine
培哚普利叔丁胺,培哚普利叔丁胺盐,S9490-3,Perindopril tert-butylamine salt |
Apoptosis; RAAS; MRP | Apoptosis; Endocrinology/Hormones; Immunology/Inflammation |
Perindopril erbumine (S9490-3) 是一种长效血管紧张素转换酶抑制剂。 | |||
T7339 |
Angiotensin (1-7)
Ang-(1-7),Angiotensin 1-7,ASP-ARG-VAL-TYR-ILE-HIS-PRO |
RAAS; Endogenous Metabolite | Endocrinology/Hormones; Metabolism |
Angiotensin (1-7) (ASP-ARG-VAL-TYR-ILE-HIS-PRO) 是肾素-血管紧张素系统中的内源性七肽。Angiotensin 1-7在心肌细胞中具有抗炎和抗纤维化活性,因此具有心脏保护作用。它能抑制血管紧张素转换酶和释放一氧化氮,是激肽诱导的血管舒张的局部协同调节剂。它阻断 Ang II 诱导的平滑肌细胞增殖和肥大,并显示对内皮的抗血管生成和生长抑制作用。它显示出抗炎活性。 | |||
T6486 |
Enalapril Maleate
MK-421 Maleate,Renitec Maleate,Glioten Maleate,MK-421 (maleate),Vasotec Maleate,马来酸依那普利 |
RAAS | Endocrinology/Hormones |
Enalapril Maleate (MK-421 Maleate) 一种是血管紧张素转化酶(ACE)抑制剂。 | |||
T6595 |
Moexipril hydrochloride
莫昔普利盐酸盐,Moexipril HCl,RS-10085,SPM 925,CI-925 |
Apoptosis; RAAS | Apoptosis; Endocrinology/Hormones |
Moexipril hydrochloride (Moexipril HCl) 是一种有口服活性的,不含巯基的血管紧张素转化酶抑制剂,可治疗高血压和充血性心力衰竭。 | |||
T6698 |
Temocapril hydrochloride
CS-622 HCl,Acecol,Temocapril HCl,CS-622,盐酸替莫普利 |
RAAS | Endocrinology/Hormones |
Temocapril hydrochloride (CS-622 HCl) 是血管紧张素转化酶 (ACE) 抑制剂。Temocapril HCl 能够用于充血性心力衰竭、急性心肌梗死、高血压、胰岛素抵抗和肾脏疾病的研究。 | |||
T6444 |
Cilazapril Monohydrate
Ro 31-2848 monohydrate,Justor,西拉普利,西拉普利水合物 |
RAAS | Endocrinology/Hormones |
Cilazapril Monohydrate (Justor) 是一种血管紧张素转化酶抑制剂,能够作用于高血压和充血性心力衰竭的研究。 | |||
T24906L |
Tuna AI acetate
|
Angiotensin-converting Enzyme (ACE) | Metabolism |
Tuna AI acetate 是一种源自金枪鱼肌肉的非竞争性血管紧张素转换酶 (ACE) 抑制剂。 | |||
TP1920L1 |
Acein acetate
|
RAAS | Endocrinology/Hormones |
Acein acetate 是高亲和力血管紧张素转换酶 (ACE) 配体 (Kd = 2.79 nM)。浓度高达 500 nM 时对 ACE 酶活性没有显着影响。增强 NMDA + D-丝氨酸诱导的多巴胺从体外纹状体切片和体内纹状体的释放。 | |||
TP1750L |
H-Ile-Pro-Pro-OH acetate
H-Ile-Pro-Pro-OH acetate(26001-32-1 free base) |
Angiotensin-converting Enzyme (ACE) | Metabolism |
H-Ile-Pro-Pro-OH acetate 是一种血管紧张素转换酶抑制剂,为乳源三肽。 | |||
TP1682L |
Abz-FR-K(Dnp)-P-OH acetate
Abz-FR-K(Dnp)-P-OH acetate (500799-61-1 free base) |
Others | Others |
Abz-FR-K(Dnp)-P-OH acetate(500799-61-1 free base) 是一种出色的血管紧张素 I 转换酶 (ACE) 底物,Km 值为 4.0 μM,kcat 值为 210s-1。 | |||
TP1404L |
Hemorphin-7 acetate(152685-85-3 free base)
|
Opioid Receptor | Endocrinology/Hormones; GPCR/G Protein; Neuroscience |
Hemorphin-7 acetate(152685-85-3 free base) 是一种 hemorphin 肽,一种源自血红蛋白 β 链的内源性阿片肽。 Hemorphin 肽具有镇痛和抗高血压活性,可激活阿片受体并抑制血管紧张素转换酶 (ACE)。 | |||
TP1917L1 |
Sar-[D-Phe8]-des-Arg9-Bradykinin acetate
Sar-[D-Phe8]-des-Arg9-Bradykinin acetate(126959-88-4 free base) |
Bradykinin Receptor | GPCR/G Protein |
Sar-[D-Phe8]-des-Arg9-Bradykinin acetate(126959-88-4 free base) 是一种有效的选择性缓激肽 B1 受体激动剂(兔主动脉中的 EC50 = 9.02 nM),对氨肽酶、激肽酶 I 和 II (ACE) 以及中性内肽酶切割具有抗性。在体内表现出降血压和血管生成活性。 | |||
T37340 |
N4-Acetylsulfamethoxazole
N-acetyl Sulfamethoxazole,醋磺胺甲噁唑 |
Others | Others |
N4-Acetylsulfamethoxazole 是磺胺甲恶唑的一种代谢物。Sulfamethoxazole 属于磺胺类抗菌素,可用于细菌感染。 | |||
T36851L |
Peptide5 acetate
|
Others | Others |
Peptide5 acetate 可减少脊髓损伤后的动物肿胀、星形胶质细胞增生和神经元细胞死亡。 Peptide5 acetate 显着降低啮齿动物离体模型中的脊髓损伤 (SCI) 程度。 | |||
T9896 |
7-Methoxy-1-naphthylacetonitrile
|
Others | Others |
7-Methoxy-1-naphthylacetonitrile 是抗抑郁药阿戈美拉汀的杂质之一。 | |||
T9269 |
N-Chloroacetyl-3,5-bis(trifluoromethyl)aniline
N1-[3,5-双(三氟甲基)苯基]-2-氯乙酰胺,N-(3,5-Bis(trifluoromethyl)phenyl)-2-chloroacetamide |
Others | Others |
N-Chloroacetyl-3,5-bis(trifluoromethyl)aniline (KM1954) 是一种杀虫剂,对第一阶段Ae 有效。 LC50 值为 125μM 的埃及伊蚊幼虫。 | |||
T17326 |
2,3,4,6-Tetra-o-acetyl-alpha-galactosylpyranosyl bromide
2-3-4-6-tetra-o-acetyl-alpha-galactosylpyranosyl-bromide |
Others; PROTAC Linker | Others; PROTAC |
2,3,4,6-Tetra-o-acetyl-alpha-galactosylpyranosyl bromide (2-3-4-6-tetra-o-acetyl-alpha-galactosylpyranosyl-bromide) 是一种属于 alkyl chain 类的 PROTAC linker,可用于 PROTAC 分子的合成。 | |||
T8368 |
Geranylacetone(Z/E)
6,10-二甲基-5,9-十一双烯-2-酮,Dihydropseudoionone |
Others | Others |
Geranylacetone(Z/E) (Dihydropseudoionone) 是一种天然存在的化合物,存在于许多植物的精油中,包括迷迭香、薰衣草和茉莉花。它具有抗氧化、抗炎和抗微生物的特性。 | |||
TP2180L |
Compstatin control peptide acetate
|
Complement System | Immunology/Inflammation |
Compstatin control peptide acetate 是补体蛋白 C3 的抑制剂,通过结合和抑制补体 C3 的切割。 | |||
T22427 |
Dehydroacetic acid sodium
脱氢醋酸钠,Sodium dehydroacetate |
Antibacterial; Antifungal | Microbiology/Virology |
Dehydroacetic acid sodium (Sodium dehydroacetate) 是一种吡喃衍生物,具有植物毒性作用,可作抗菌和抗真菌剂。 | |||
T78230 |
2,4′-Dichloroacetanilide
2-chloro-N-(4-chlorophenyl)acetamide |
Others | Others |
2,4′-Dichloroacetanilide (2-chloro-N-(4-chlorophenyl)acetamide) 具有抗真菌活性,抑制 T. asteroides,其最小抑菌浓度为 6.25 μg/mL。 | |||
T1608 |
ADH-1 trifluoroacetate
Exherin trifluoroacetate |
Dehydrogenase | Metabolism |
ADH-1 trifluoroacetate (Exherin trifluoroacetate) 是一种选择性的、竞争性N-钙粘蛋白拮抗剂,具有潜在抗肿瘤和抗血管生成作用。 | |||
T17330 |
2-Phthalimidehydroxy-acetic acid
|
Others; PROTAC Linker | Others; PROTAC |
2-Phthalimidehydroxy-acetic acid 是一种属于 alkyl chain 类的 PROTAC linker,可用于 PROTAC 分子的合成。 | |||
T9944 |
3-(9-Chloro-3-methyl-4-oxoisoxazolo[4,3-c]quinolin-5(4H)-yl)-N-(3,4,5-trimethoxyphenyl)benzeneacetamide
|
MRP | Immunology/Inflammation |
3-(9-Chloro-3-methyl-4-oxoisoxazolo[4,3-c]quinolin-5(4H)-yl)-N-(3,4,5-trimethoxyphenyl)benzeneacetamide inhibits multidrug resistance protein (MRP1). |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T5S0106 |
Peimisine
贝母辛,Ebeiensine |
RAAS; AChR | Endocrinology/Hormones; Neuroscience |
Peimisine (Ebeiensine) 非竞争性拮抗气管平滑肌 M 受体,抑制 Ach 引起的平滑肌收缩。它兴奋 β 受体和拮抗内钙释放,促进一氧化氮释放,可舒张气管平滑肌,有平喘作用。 | |||
T13299 |
Vicenin 3
维采宁-3,维采宁 3 |
RAAS | Endocrinology/Hormones |
Vicenin 3来源于广金钱草的地上部分。Vicenin 3是血管紧张素转换酶抑制剂,IC50=46.91 μM。 | |||
T8270 |
Deserpidine
地舍平,Harmonyl |
RAAS | Endocrinology/Hormones |
Deserpidine (Harmonyl) 是从 Rauwolfia canescens 的根中分离的生物碱。Deserpidine 与 Reserpine 相关。Deserpidine 是竞争性血管紧张素转化酶抑制剂,可以被用作抗高血压药以及镇定剂。Deserpidine 还减少了肾上腺皮质血管紧张素 II 诱导的醛固酮分泌。 | |||
T5796 |
Plantainoside D
Isoplantamajoside,车前草苷D |
RAAS; PKC | Chromatin/Epigenetic; Cytoskeletal Signaling; Endocrinology/Hormones |
Plantainoside D (Isoplantamajoside) 可以抑制 ACE ,IC50=2.17 mM。Plantainoside D 也是IKK-β抑制剂。 | |||
T21418 |
Lisinopril
Linopril,赖诺普利,Zestril,Prinivil,Lisipril |
RAAS | Endocrinology/Hormones |
Lisinopril (Prinivil) 是一种血管紧张素转化酶抑制剂,能够作用于高血压,充血性心力衰竭和心脏病等。 | |||
T3851 |
Vicenin 2
Vicenin -2,维采宁 2,新西兰牡荆苷 |
RAAS | Endocrinology/Hormones |
Vicenin 2 来源于广金钱草 (Desmodium styracifolium) 的地上部分。Vicenin 2 是一种血管紧张素转换酶 (ACE) 抑制剂,IC50=43.83 μM。 | |||
T3753 |
Sinapinic Acid
Sinapic acid,芥子酸,Synapoic acid |
Apoptosis; RAAS; Reactive Oxygen Species; HDAC | Apoptosis; Chromatin/Epigenetic; DNA Damage/DNA Repair; Endocrinology/Hormones; Immunology/Inflammation; Metabolism; NF-κB |
Sinapinic Acid (Synapoic acid) 是从 Hydnophytum formicarumJack. 根中分离到的酚类,是HDAC 抑制剂,对ACE-I 的活性也有抑制作用。它有抗肿瘤活性,诱导肿瘤细胞凋亡,具有抗氧化、抗糖尿病的作用。 | |||
T6627 |
Phosphoramidon Disodium
Phosphoramidon Disodium Salt,磷酰胺二钠 |
RAAS; Neprilysin; Others | Endocrinology/Hormones; Metabolism; Others |
Phosphoramidon Disodium (Phosphoramidon Disodium Salt) Salt 是一种金属蛋白酶 (metalloprotease) 抑制剂 。Phosphoramidon Disodium Salt 抑制内皮素转化酶 (ECE) ,中性肽内切酶 (NEP) 和血管紧张素转换酶 (ACE) 的IC50分别为 3.5 ,0.034 和 78 μM。 | |||
T67047 |
2-Acetyl-3-ethylpyrazine
|
Endogenous Metabolite | Metabolism |
2-Acetyl-3-ethylpyrazine 具有抗肿瘤活性。 | |||
T5132 |
9-dihydro-13-acetylbaccatin III
13-乙酰基-9-羟基巴卡丁 III,13-Acetyl-9-dihydrobaccatin III,9-DHAB III |
Apoptosis | Apoptosis |
9-dihydro-13-acetylbaccatin III (9-DHAB III) 是一种制备紫杉醇类似物的中间体。 | |||
T8059 |
N-Acetyl-L-methionine
N-Acetylmethionine,N-乙酰-L-蛋氨酸 |
Others; Endogenous Metabolite | Metabolism; Others |
N-Acetyl-L-methionine (N-Acetylmethionine) 是人体代谢物,在营养和代谢作用上和 L-methionine 相当。其中 L-methionine 是生长发育并不能够少的氨基酸。 | |||
T4456 |
N4-Acetylcytidine
N4-乙酰胞苷,N-Acetylcytidine |
Others; Endogenous Metabolite | Metabolism; Others |
N4-Acetylcytidine (N-Acetylcytidine) 是内源性代谢产物的一种。 | |||
T7299 |
β-Estradiol 17-acetate
β-雌二醇 17-乙酸酯,17-乙酸-17-BETA-雌二酯,beta-estradiol 17-acetate,1,3,5(10)-Estratriene-3,17β-diol 17-acetate |
Estrogen Receptor/ERR; Others | Endocrinology/Hormones; Others |
β-Estradiol 17-acetate (1,3,5(10)-Estratriene-3,17β-diol 17-acetate) 是一种雌二醇代谢物。 | |||
T5145 |
Oxytocin acetate
Oxytocic hormone acetate,α-Hypophamine acetate,Oxytocin acetate (50-56-6 free base),醋酸催产素 |
Oxytocin Receptor | Endocrinology/Hormones; GPCR/G Protein |
Oxytocin acetate (α-Hypophamine acetate) 是哺乳动物的神经垂体激素,是多效的下丘脑肽,是催产素受体的配体,有助于分娩、哺乳和亲社会行为。它可作为一种压力应对分子,具有抗炎、抗氧化剂和保护作用。 | |||
T3751 |
2',4'-Dihydroxyacetophenone
Resacetophenone,雷琐乙酰苯,1-(2,4-Dihydroxyphenyl)ethanone,2,4-Dihydroxyacetophenone,4-Acetylresorcinol |
Others; Endogenous Metabolite | Metabolism; Others |
2',4'-Dihydroxyacetophenone (Resacetophenone) 是一种植物代谢物,是在2'和4'位置被羟基取代基的苯乙酮。。 | |||
T41122 |
1,3-Dihydroxyacetone
|
Endogenous Metabolite | Metabolism |
1,3-Dihydroxyacetone 是防晒美黑护肤制剂的主要活性成分,是合成各种精细化学品的重要前体,也是一种食品添加剂,可通过在 Gluconobacter oxydans 上进行微生物发酵实现工业规模生产。1,3-Dihydroxyacetone 具有提高cAMP 水平的能力。 | |||
TN7158 |
2-(4-methoxyphenyl)-N-methyl-2-oxoacetamide
N-Methyl-2-(4-methoxyphenyl)-2-oxoacetamide,2-(4-methoxy-phenyl)-N-methyl-2-oxo-acetamide |
Others | Others |
2-(4-methoxyphenyl)-N-methyl-2-oxoacetamide (2-(4-methoxy-phenyl)-N-methyl-2-oxo-acetamide) 是一种海洋来源的天然产物,存在于Polycarpa aurata。 | |||
T0065 |
Acetaminophen
对乙酰氨基酚,醋氨酚,4-Acetamidophenol,4'-Hydroxyacetanilide,APAP,Paracetamol |
COX; Endogenous Metabolite; Histone Acetyltransferase | Chromatin/Epigenetic; Immunology/Inflammation; Metabolism; Neuroscience |
Acetaminophen (APAP) 是一种 COX 抑制剂,抑制 COX-1 和 COX-2 (IC50=113.7/25.8 μM)。Acetaminophen 具有解热镇痛活性,以及较弱的抗炎活性。 | |||
TN1499 |
Cimiracemoside C
千层纸素A-7-0-Β-D-葡萄糖醛酸苷,Cimicifugoside M |
AMPK | Chromatin/Epigenetic; PI3K/Akt/mTOR signaling |
Cimiracemoside C (Cimicifugoside M) 是在升麻中发现的一种天然产物,可激活 AMPK 并具有抗糖尿病的潜在活性。 | |||
TN4417 |
Larixyl acetate
|
Others | Others |
Larixyl acetate 是一种生物活性化学物质。 | |||
T2956 |
Cedryl acetate
乙酸柏木酯,Cedrol acetate,Cedranyl acetate |
Antifungal | Microbiology/Virology |
Cedryl acetate (Cedranyl acetate) 是一种三环倍半萜烯,分离自草莓番石榴植物,能够表现出 α-葡萄糖苷酶的抑制活性。 | |||
TN6773 |
Acetoxyvalerensre
acetylvalerenolic acid |
GABA Receptor | Membrane transporter/Ion channel; Neuroscience |
Acetoxyvalerensre (acetylvalerenolic acid) 是缬草酸的衍生物,它是一种 GABAA 受体调节剂。 | |||
T8088 |
Furfuryl acetate
乙酸糠醇酯,乙酸糠酯 |
Others | Others |
Furfuryl acetate 可用于合成 5-乙酰氧基甲基-2-呋喃和 5-羟甲基-2-呋喃。 | |||
T5S2245 |
Alisol C 23-acetate
泽泻醇 C-23-醋酸酯,Alisol C monoacetate |
Others | Others |
Alisol C 23-acetate (Alisol C monoacetate) 是一种提取自东方泽泻中的天然产物,可以显著减少迟发型超敏反应。 | |||
T8024 |
3-Indoleacetonitrile
|
Others; Endogenous Metabolite | Metabolism; Others |
3-Indoleacetonitrile 是内源性代谢产物的一种。 | |||
TQ0099 |
20-O-Acetylingenol-3-angelate
巨大戟醇-3-O-当归酸-20-乙酸酯,Euphorbia factor Pe1 |
Others | Others |
20-O-Acetylingenol-3-angelate (Euphorbia factor Pe1) 是一种天然化合物,存在于植物英加的叶子和茎中。它具有多种生物活性,包括抑制肿瘤生长、抗炎、抗真菌和抗氧化作用。 | |||
T1273 |
Diacerein
双醋瑞因,Diacerhein,Fisiodar,Diacetylrhein |
IL Receptor; Interleukin | Immunology/Inflammation |
Diacerein (Fisiodar) 是一种慢效具有白介素-1β 抑制效果的蒽醌类化合物。 | |||
T8160 |
EGCG Octaacetate
乙酰化表没食子儿茶素没食子酸酯,乙酰化EGCG |
Others; Antibacterial | Microbiology/Virology; Others |
EGCG Octaacetate 是表没食子儿茶素没食子酸酯的前药,对革兰氏阳性菌和革兰氏阴性菌有潜在抗菌可能。它可下调 PI3K/Akt/NFκB 磷酸化和 p65 乙酰化来降低促炎介质水平,减少小鼠结肠炎引起的结肠癌。 | |||
TN3340 |
Acetylatractylodinol
Tractylodinol acetate,乙酰基仓术呋喃烃醇 |
Others | Others |
Acetylatractylodinol (Tractylodinol acetate) 是分离自Atractylodes lancea 中,具有抗氧化作用。 | |||
T8168 |
Hydroxytyrosol Acetate
3,4-二羟基苯乙醇醋酸,HTy-Ac |
Antioxidant | oxidation-reduction |
Hydroxytyrosol Acetate (HTy-Ac) 是从橄榄油中发现的,具有抗氧化作用。它清除 DPPH 自由基的活性比 hydroxytyrosol 弱。 | |||
T0269 |
Dichlorisone Acetate
糊状叶绿素,Diloderm,醋酸二氯松 |
Endogenous Metabolite; AChE | Metabolism; Neuroscience |
Dichlorisone Acetate (Diloderm) 一种是合成的糖皮质激素皮质类固醇,具有抗炎特性。 | |||
T5S2357 |
Acetylcorynoline
(+)-Corynoline Acetate,O-Acetylcorynoline,乙酰紫堇灵 |
Antifungal | Microbiology/Virology |
Acetylcorynoline (O-Acetylcorynoline) 是提取自 Corydalis bungeana 中的一种主要生物碱成分,具有抗炎活性。 | |||
T15254 |
Ethyl acetoacetate
Ethyl acetylacetate |
Others; Antibacterial | Microbiology/Virology; Others |
Ethyl acetoacetate (Ethyl acetylacetate) 是一种细菌生物膜抑制剂。Ethyl acetoacetate 是一种酯类,是一种可用于多种化合物合成的中间体。 | |||
TMA0536 |
2-Acetylbenzoic acid
|
Prostaglandin Receptor | GPCR/G Protein; Immunology/Inflammation |
2-Acetylbenzoic acid 在抑制血小板功能和血小板前列腺素 (PG) 合成方面比 2-丙酰氧基苯甲酸更有效,尽管这些药物在抑制前列环素 (PGI2) 合成方面的效力相当。 | |||
TQ0316 |
Ingenol-5,20-acetonide-3-O-angelate
Ingenol 5,20-acetonide 3-angelate,Ingenol 3-angelate 5,20-acetonide,巨大戟醇-5,20-缩丙酮-3-当归酸酯 |
Others | Others |
Ingenol-5,20-acetonide-3-O-angelate (Ingenol 5,20-acetonide 3-angelate) 是一种天然产物。 | |||
T3750 |
4-Hydroxyacetophenone
对羟基苯乙酮,4-Acetylphenol,Piceol,p-Acetylphenol,4'-Hydroxyacetophenone |
HBV; Xanthine Oxidase | Metabolism; Microbiology/Virology |
4-Hydroxyacetophenone (4-Acetylphenol) 是蒿属植物和木香属植物中的一种黄嘌呤氧化酶抑制剂,具有保肝促胆、抗乙型肝炎病毒和抗炎作用。 | |||
T1284 |
Megestrol acetate
SC10363,醋酸甲地孕酮,BDH1298 |
Glucocorticoid Receptor; Estrogen/progestogen Receptor; Progesterone Receptor; HIV Protease; Autophagy | Autophagy; Endocrinology/Hormones; Microbiology/Virology; Others; Proteases/Proteasome |
Megestrol acetate (BDH1298) 是具有口服活性的合成孕激素。它还具有抗雄激素特性,可用于治疗厌食症和恶病质。 | |||
T20587 |
2-Acetonaphthone
2-萘乙酮,beta-Acetylnaphthalene,beta-Acetonaphthalene,2Acetylnaphthalene,2-Acetylnaphthalene,2 Acetylnaphthalene,beta-Naphthyl methyl ketone |
Endogenous Metabolite | Metabolism |
2-Acetonaphthone (beta-Naphthyl methyl ketone) 是内源性代谢产物的一种。 | |||
T4S2014 |
5,15-Diacetyl-3-benzoyllathyrol
,大戟因子L3,二乙酰基苯甲酰基香豌豆醇,5,15-二乙酰基-3-苯甲酰千金子二萜醇;千金二萜醇二乙酰苯甲酰酯,Euphorbia factor L3 |
Others | Others |
5,15-Diacetyl-3-benzoyllathyrol (Euphorbia factor L3) 是一种具有抗癌作用的萜类化合物。 | |||
T1016 |
D-α-Tocopherol acetate
乙酸维生素E,Vitamin E Acetate,Tocopherol acetate |
Endogenous Metabolite | Metabolism |
D-α-Tocopherol acetate (Vitamin E Acetate) 能够水解为 d-α-生育酚 (VE) 并被小肠吸收。 | |||
Fr12596 |
3-Acetylcoumarin
|
Others | Others |
3-Acetylcoumarin 作为室温下铜催化 CN 偶联反应的实用配体。它具有神经保护和杀螨特性。 | |||
T4907 |
3,4-Dihydroxybenzeneacetic acid
DOPAC,3,4-Dihydroxyphenylacetic acid,3,4-二羟基苯乙酸 |
Endogenous Metabolite | Metabolism |
3,4-Dihydroxybenzeneacetic acid (3,4-Dihydroxyphenylacetic acid) 是一种多巴胺的主要神经元代谢产物。 | |||
T3819 |
Ursolic acid acetate
熊果酸乙酸酯,Acetylursolic acid,3-Acetylursolic Acid |
AChE | Neuroscience |
Ursolic acid acetate (Acetylursolic acid) 分离于 Ficus microcarpa 的气根中,对 KB 细胞显示细胞毒性(IC50:8.4 μM)。 | |||
T6S2246 |
Alisol B 23-acetate
Alisol B Acetate,Alisol B monoacetate,23-O-Acetylalisol B,23-Acetylalismol B,泽泻醇B乙酸酯 |
Others | Others |
Alisol B 23-acetate (Alisol B Acetate) 是三萜类化合物,能够激活法尼醇受体,诱导受损的肝脏再生。 | |||
T9780 |
3,4, 5-trimethoxyphenylacetic acid
|
Endogenous Metabolite | Metabolism |
3,4, 5-trimethoxyphenylacetic acid 是有机合成中常见的中间体,其主要用途是将其羧基转化为相应的用途。 | |||
TN6710 |
Methyl acetylsalicylate
ACETYLSALICYLIC ACID METHYL ESTER,乙酰水杨酸甲酯 |
Others | Others |
Methyl acetylsalicylate (ACETYLSALICYLIC ACID METHYL ESTER) 是一种从豌豆中分离出来的天然产物。抑制胶原蛋白诱导的人富含血小板的血浆聚集。 | |||
T4946 |
(+)-Columbianetin acetate
二氢欧山芹醇醋酸酯,COLUMBIANETIN ACETATE |
Others | Others |
(+)-Columbianetin acetate (COLUMBIANETIN ACETATE) 是一种 Columbianetin 异构体。其中Columbianetin 是植物抗毒素,与芹菜贮藏过程中对病原体的抗性有关,表现出良好的抗炎及抗真菌活性。 | |||
T3033 |
Deoxycorticosterone acetate
醋酸去氧皮质酮,DOC acetate,Cortexone acetate,11-Deoxycorticosterone acetate,醋酸脱氧皮质酮 |
Glucocorticoid Receptor; Endogenous Metabolite; Adrenergic Receptor | Endocrinology/Hormones; GPCR/G Protein; Metabolism; Neuroscience |
Deoxycorticosterone acetate (Cortexone acetate) 是肾上腺产生的类固醇激素,具有盐皮质激素活性,并作为醛固酮的前体。 | |||
TN7190 |
3-Bromo-4-Methoxyphenylacetonitrile
3-Bromo-4-methoxybenzyl Cyanide,ZINC2565991,2-(3-bromo-4-methoxyphenyl)acetonitrile,3-溴-4-甲氧基苯乙腈 |
Others | Others |
3-Bromo-4-Methoxyphenylacetonitrile (ZINC2565991) 是一种海洋来源的天然产物,存在于 Aiolochroia crassa。 | |||
TN1149 |
6''-O-acetylsaikosaponin A
|
Others | Others |
6''-O-Acetylsaikosaponin A 是一种分离自柴胡根中的乙酰柴胡皂苷,表现出一定的破骨细胞抑制活性。 | |||
------------------------ 更多 ------------------------ |
Cat. No. | Product Name | Species | Expression System |
---|---|---|---|
TMPK-00383 |
ACE2/ACEH Protein, Human, Recombinant (His & Avi)
ACE2,ACE-2,ACEH |
Human | HEK293 Cells |
ACE2 (Angiotensin I Converting Enzyme 2) is a Protein Coding gene. Diseases associated with ACE2 include Severe Acute Respiratory Syndrome and Neurogenic Hypertension.The protein encoded by this gene belongs to the angiotensin-converting enzyme family of dipeptidyl carboxydipeptidases and has considerable homology to human angiotensin 1 converting enzyme. This secreted protein catalyzes the cleavage of angiotensin I into angiotensin 1-9, and angiotensin II into the vasodilator angiotensin 1-7. A... | |||
TMPK-00382 |
ACE2/ACEH Protein, Human, Recombinant (hFc & Avi), Biotinylated
ACE-2,ACE2,ACEH |
Human | HEK293 Cells |
ACE2 (Angiotensin I Converting Enzyme 2) is a Protein Coding gene. Diseases associated with ACE2 include Severe Acute Respiratory Syndrome and Neurogenic Hypertension.The protein encoded by this gene belongs to the angiotensin-converting enzyme family of dipeptidyl carboxydipeptidases and has considerable homology to human angiotensin 1 converting enzyme. This secreted protein catalyzes the cleavage of angiotensin I into angiotensin 1-9, and angiotensin II into the vasodilator angiotensin 1-7. A... | |||
TMPK-00551 |
ACE2/ACEH Protein, Cynomolgus, Recombinant (His & Avi)
ACE-2,ACEH,ACE2 |
Cynomolgus | HEK293 Cells |
ACE2 (Angiotensin I Converting Enzyme 2) is a Protein Coding gene. Diseases associated with ACE2 include Severe Acute Respiratory Syndrome and Neurogenic Hypertension.The protein encoded by this gene belongs to the angiotensin-converting enzyme family of dipeptidyl carboxydipeptidases and has considerable homology to human angiotensin 1 converting enzyme. This secreted protein catalyzes the cleavage of angiotensin I into angiotensin 1-9, and angiotensin II into the vasodilator angiotensin 1-7. A... | |||
TMPK-00552 |
ACE2/ACEH Protein, Cynomolgus, Recombinant (His & Avi), Biotinylated
ACEH,ACE-2,ACE2 |
Cynomolgus | HEK293 Cells |
ACE2 (Angiotensin I Converting Enzyme 2) is a Protein Coding gene. Diseases associated with ACE2 include Severe Acute Respiratory Syndrome and Neurogenic Hypertension.The protein encoded by this gene belongs to the angiotensin-converting enzyme family of dipeptidyl carboxydipeptidases and has considerable homology to human angiotensin 1 converting enzyme. This secreted protein catalyzes the cleavage of angiotensin I into angiotensin 1-9, and angiotensin II into the vasodilator angiotensin 1-7. A... | |||
TMPJ-00386 |
ACE2/ACEH Protein, Human, Recombinant (HEK293, His & Avi), Biotinylated
Metalloprotease MPROT15,ACEH,Angiotensin-Converting... |
Human | HEK293 Cells |
Angiotensin-Converting Enzyme 2 (ACE-2) is an integral membrane protein and a zinc metalloprotease of the ACE family, the ACE family includes somatic and germinal ACE. ACE-2 cleaves angiotensins I and II as a carboxypeptidase, ACE-2 converts angiotensin I to angiotensin 1-9, and angiotensin II to angiotensin 1-7. ACE-2 is also able to hydrolyze apelin-13 and dynorphin-13 with high efficiency. ACE-2 can be high expressed in testis, kidney and heart, in colon, small intestine and ovary at moderate... | |||
TMPH-03081 |
ACE2 Protein, Paguma larvata, Recombinant (hFc)
EC:3.4.17.23,Angiotensin-converting enzyme 2,ACE-re... |
Paguma larvata | HEK293 Cells |
ACE2 Protein, Paguma larvata, Recombinant (hFc) is expressed in HEK293 mammalian cells with C-hFc tag. The predicted molecular weight is 112.7 kDa and the accession number is Q56NL1. | |||
TMPY-02207 |
ACE2/ACEH Protein, Rat, Recombinant (His)
angiotensin I converting enzyme 2 |
Rat | HEK293 Cells |
ACE2/ACEH Protein, Rat, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 85 kDa and the accession number is Q5EGZ1. | |||
TMPY-01838 |
ACE2/ACEH Protein, Mouse, Recombinant (His)
angiotensin I converting enzyme 2,2010305L05Rik |
Mouse | HEK293 Cells |
ACE2/ACEH Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 85 kDa and the accession number is Q8R0I0-1. | |||
TMPY-01839 |
ACE2/ACEH Protein, Mouse, Recombinant (His & hFc)
2010305L05Rik,angiotensin I converting enzyme 2 |
Mouse | HEK293 Cells |
ACE2/ACEH Protein, Mouse, Recombinant (His & hFc) is expressed in HEK293 mammalian cells with His and hFc tag. The predicted molecular weight is 112 kDa and the accession number is Q8R0I0-1. | |||
TMPY-03561 |
ACE2/ACEH Protein, Rhesus, Recombinant (hFc)
angiotensin I converting enzyme 2 |
Rhesus | HEK293 Cells |
ACE2/ACEH Protein, Rhesus, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 110.7kDa and the accession number is B6DUF3. | |||
TMPY-03830 |
ACE2/ACEH Protein, Rhesus, Recombinant (His)
angiotensin I converting enzyme 2 |
Rhesus | HEK293 Cells |
ACE2/ACEH Protein, Rhesus, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 85.1 kDa and the accession number is B6DUF3. | |||
TMPY-04312 |
ACE2/ACEH Protein, Human, Recombinant (mFc)
angiotensin I converting enzyme 2,ACEH |
Human | HEK293 Cells |
ACE2/ACEH Protein, Human, Recombinant (mFc) is expressed in HEK293 mammalian cells with mFc tag. The predicted molecular weight is 110 kDa and the accession number is Q9BYF1-1. | |||
TMPY-05266 |
ACE2/ACEH Protein, Human, Recombinant (His)
ACEH,angiotensin I converting enzyme 2 |
Human | HEK293 Cells |
ACE2/ACEH Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 85.1 kDa and the accession number is Q9BYF1-1. | |||
TMPY-06334 |
ACE2/ACEH Protein, Human, Recombinant (hFc), Biotinylated
ACEH,angiotensin I converting enzyme 2 |
Human | HEK293 Cells |
ACE2/ACEH Protein, Human, Recombinant (hFc), Biotinylated is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 110.3 kDa and the accession number is NP_068576.1. | |||
TMPY-00655 |
ACE2/ACEH Protein, Human, Recombinant (hFc)
angiotensin I converting enzyme 2,ACEH |
Human | HEK293 Cells |
ACE2/ACEH Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 110.3 kDa and the accession number is Q9BYF1-1. | |||
TMPY-05725 |
ACE2/ACEH Protein, Human, Recombinant (His & Avi), Biotinylated
angiotensin I converting enzyme 2,ACEH |
Human | Baculovirus Insect Cells |
ACE2/ACEH Protein, Human, Recombinant (His & Avi), Biotinylated is expressed in Baculovirus insect cells with His and Avi tag. The predicted molecular weight is 86.86 kDa and the accession number is Q9BYF1-1. | |||
TMPY-05696 |
ACE2/ACEH Protein, Human, Recombinant (His), Biotinylated
ACEH,angiotensin I converting enzyme 2 |
Human | HEK293 Cells |
ACE2/ACEH Protein, Human, Recombinant (His), Biotinylated is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 85.1 kDa and the accession number is Q9BYF1-1. | |||
TMPY-00678 |
BACE1 Protein, Mouse, Recombinant (His)
beta-site APP-cleaving enzyme 1,C76936,β-site APP-cleaving e... |
Mouse | HEK293 Cells |
BACE1 Protein, Mouse, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 49.8 kDa and the accession number is P56818. | |||
TMPY-03065 |
BACE2 Protein, Mouse, Recombinant (His)
CEAP1,BAE2,1110059C24Rik,β-site APP-cleaving enzyme 2,CDA13,... |
Mouse | HEK293 Cells |
BACE2, also known as beta secretase 2, belongs to the peptidase A1 family. It is a protease known to be an important enzyme involved in the cellular pathways. BACE2 has been shown to interact with GGA1 and GGA2. It is the major β-secretase in vivo. BACE2 is located on chromosome 21 and may play a role in alzheimer's disease pathogenesis in down syndrome(DS). Overexpression of BACE2 by lentivirus markedly reduced amyloid β protein production in primary neurons. Despite an extra copy of the BACE2 ... | |||
TMPH-03234 |
Acetylcholinesterase Protein, Rat, Recombinant (His)
AChE,EC:3.1.1.7 |
Rat | E. coli |
Terminates signal transduction at the neuromuscular junction by rapid hydrolysis of the acetylcholine released into the synaptic cleft. Acetylcholinesterase Protein, Rat, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 68.9 kDa and the accession number is P37136. | |||
TMPH-02464 |
AIIM Protein, Microbacterium testaceum, Recombinant (His & SUMO)
AHL-lactonase,N-acyl homoserine lactonase |
Microbacterium testaceum | E. coli |
Hydrolyzes short- and long-chain N-acyl homoserine lactones with or without 3-oxo substitution at C3. Has slight activity towards L-homoserine lactone, and no activity towards gamma-butyrolactone. AIIM Protein, Microbacterium testaceum, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 43.3 kDa and the accession number is C6L862. | |||
TMPH-00339 |
Acetyl-CoA carboxylase Protein, Candida glabrata, Recombinant (His)
ACC1 |
Candida glabrata | E. coli |
Acetyl-CoA carboxylase Protein, Candida glabrata, Recombinant (His) is expressed in E. coli expression system with N-10xHis tag. The predicted molecular weight is 67.2 kDa and the accession number is A0A0W0CTK3. | |||
TMPH-00051 |
Chitin deacetylase Protein, Amylomyces rouxii, Recombinant (His)
Chitin deacetylase,MrCDA,CDA |
Amylomyces rouxii | E. coli |
Hydrolyzes the N-acetamido groups of N-acetyl-D-glucosamine residues in chitin to form chitosan and acetate. Chitin deacetylase Protein, Amylomyces rouxii, Recombinant (His) is expressed in E. coli expression system with N-10xHis tag. The predicted molecular weight is 49.9 kDa and the accession number is P50325. | |||
TMPY-00107 |
Influenza A H18N11 (A/flat-faced bat/Peru/033/2010) Hemagglutinin/HA1 Protein (His)
Harvey rat sarcoma viral oncogene homolog |
H18N11 | HEK293 Cells |
Influenza A H18N11 (A/flat-faced bat/Peru/033/2010) Hemagglutinin/HA1 Protein (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 37.8 kDa and the accession number is U5N1D3. | |||
TMPY-03569 |
Betacellulin Protein, Human, Recombinant (hFc)
betacellulin,βcellulin |
Human | HEK293 Cells |
Betacellulin Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 36 kDa and the accession number is P35070. | |||
TMPY-01323 |
Betacellulin Protein, Mouse, Recombinant (His & hFc)
Bcn,betacellulin,βcellulin |
Mouse | HEK293 Cells |
Betacellulin Protein, Mouse, Recombinant (His & hFc) is expressed in HEK293 mammalian cells with His and hFc tag. The predicted molecular weight is 38 kDa and the accession number is Q05928. | |||
TMPY-06597 |
Betacellulin Protein, Rhesus, Recombinant (hFc)
betacellulin,βcellulin |
Rhesus | HEK293 Cells |
Betacellulin Protein, Rhesus, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 36 kDa and the accession number is XP_001101880.3. | |||
TMPH-00405 |
Acyl-CoA dehydrogenase Protein, Clostridium acetobutylicum, Recombinant (His & Myc)
Acyl-CoA dehydrogenase, short-chain specific,SCAD,Butyryl-Co... |
Clostridium acetobutylicum | E. coli |
Acyl-CoA dehydrogenase Protein, Clostridium acetobutylicum, Recombinant (His & Myc) is expressed in E. coli. | |||
TMPY-00652 |
BACE1 Protein, Human, Recombinant
BACE,HSPC104,β-site APP-cleaving enzyme 1,beta-site... |
Human | HEK293 Cells |
BACE1 Protein, Human, Recombinant is expressed in HEK293 mammalian cells. The predicted molecular weight is 49 kDa and the accession number is A0A024R3D7. | |||
TMPY-05019 |
Pla a 2 Protein, Platanus acerifolia, Recombinant (His)
|
Platanus acerifolia | HEK293 Cells |
PLA A2 Protein, Platanus acerifolia, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 40.7 kDa and the accession number is Q6H9K0.1. | |||
TMPH-00330 |
Acetyl-CoA carboxylase Protein, Candida albicans, Recombinant (His)
ACC1 |
Candida albicans | E. coli |
Acetyl-CoA carboxylase Protein, Candida albicans, Recombinant (His) is expressed in E. coli expression system with N-10xHis tag. The predicted molecular weight is 67.3 kDa and the accession number is A0A1D8PRR7. | |||
TMPH-03604 |
Phosphinothricin N-acetyltransferase Protein, Streptomyces hygroscopicus, Recombinant (His)
Phosphinothricin-resistance protein,Phosphinothricin N-a... |
Streptomyces hygroscopicus | E. coli |
Inactivates phosphinothricin (PPT) by transfer of an acetyl group from acetyl CoA. Can also acetylate demethylphosphinothricin but not PTT or glutamate. This enzyme is an effector of phosphinothricin tripeptide (PTT or bialaphos) resistance. Phosphinothricin N-acetyltransferase Protein, Streptomyces hygroscopicus, Recombinant (His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 24.6 kDa and the accession number is P16426. | |||
TMPH-03608 |
Phosphinothricin N-acetyltransferase Protein, S. viridochromogenes, Recombinant (His)
Phosphinothricin N-acetyltransferase,Phosphinothric... |
Streptomyces viridochromogenes | P. pastoris (Yeast) |
Inactivates phosphinothricin (PPT) by transfer of an acetyl group from acetyl CoA. This enzyme is an effector of phosphinothricin tripeptide (PTT or bialaphos) resistance. Phosphinothricin N-acetyltransferase Protein, S. viridochromogenes, Recombinant (His) is expressed in yeast with N-6xHis tag. The predicted molecular weight is 22.6 kDa and the accession number is Q57146. | |||
TMPH-03513 |
Plastocyanin Protein, Spinacia oleracea, Recombinant (His & SUMO)
Plastocyanin, chloroplastic,PETE |
Spinacia oleracea | E. coli |
Participates in electron transfer between P700 and the cytochrome b6-f complex in photosystem I. Plastocyanin Protein, Spinacia oleracea, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 26.4 kDa and the accession number is P00289. | |||
TMPY-01684 |
Placental Lactogen/CSH1 Protein, Human, Recombinant (His)
CSA,PL,CS-1,chorionic somatomammotropin hormone 1 (place... |
Human | HEK293 Cells |
Placental Lactogen/CSH1 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 23.7 kDa and the accession number is A8K6C2. | |||
TMPY-01742 |
Acetylcholinesterase Protein, Mouse, Recombinant (His)
Acre,Chrne,acetylcholinesterase (Yt blood group) |
Mouse | HEK293 Cells |
Acetylcholinesterase, also known as ACHE, is an enzyme that degrades (through its hydrolytic activity) the neurotransmitter acetylcholine, producing choline and an acetate group. Acetylcholinesterase plays a crucial role in nerve impulse transmission at cholinergic synapses by rapid hydrolysis of the neurotransmitter acetylcholine (ACh). ACHE appears to be a potential therapeutic target at muscle injuries including organophosphate myopathy. It is an externally oriented membrane-bound enzyme and ... | |||
TMPK-01326 |
Alkaline Phosphatase (Placental type) /ALPP Protein, Cynomolgus, Recombinant (His)
Alkaline phosphatase,PLAP,PLAP-1,ALPP |
Cynomolgus | HEK293 Cells |
Alkaline phosphatase can be considered "our favorite enzyme" for reasons apparent to those who diagnose and treat metabolic bone diseases or who study skeletal biology. Few might know, however, that alkaline phosphatase likely represents the most frequently assayed enzyme in all of medicine. Elevated activity in the circulation is universally recognized as a marker for skeletal or hepatobiliary disease. Alkaline Phosphatase (Placental type) /ALPP Protein, Cynomolgus, Recombinant (His) is express... | |||
TMPH-00404 |
Acetoacetate decarboxylase Protein, Clostridium acetobutylicum, Recombinant (His)
AADase,EC:4.1.1.4,ADC,AAD |
Clostridium acetobutylicum | Baculovirus Insect Cells |
Catalyzes the conversion of acetoacetate to acetone and carbon dioxide. Acetoacetate decarboxylase Protein, Clostridium acetobutylicum, Recombinant (His) is expressed in Baculovirus insect cells with C-6xHis tag. The predicted molecular weight is 33.2 kDa and the accession number is P23670. | |||
TMPH-03077 |
CGTases Protein, Paenibacillus macerans, Recombinant (E. coli, His)
CGTase,Cyclomaltodextrin glucanotransferase,Cyclodextrin-gly... |
Paenibacillus macerans | E. coli |
N/A. CGTases Protein, Paenibacillus macerans, Recombinant (E. coli, His) is expressed in E. coli expression system with N-6xHis tag. The predicted molecular weight is 15.4 kDa and the accession number is P31835. | |||
TMPH-02083 |
Serine racemase/SRR Protein, Human, Recombinant (His & SUMO)
L-serine ammonia-lyase,D-serine ammonia-lyase,Serine rac... |
Human | E. coli |
Serine racemase/SRR Protein, Human, Recombinant (His & SUMO) is expressed in E. coli. | |||
TMPH-00016 |
Ferredoxin Protein, Acetoanaerobium sticklandii, Recombinant (His & Myc)
Ferredoxin |
Acetoanaerobium sticklandii | E. coli |
Ferredoxins are iron-sulfur proteins that transfer electrons in a wide variety of metabolic reactions. | |||
TMPH-03609 |
Phosphinothricin N-acetyltransferase Protein, S. viridochromogenes, Recombinant (His & SUMO)
pat,Phosphinothricin N-acetyltransferase,Phosphinot... |
Streptomyces viridochromogenes | E. coli |
Inactivates phosphinothricin (PPT) by transfer of an acetyl group from acetyl CoA. This enzyme is an effector of phosphinothricin tripeptide (PTT or bialaphos) resistance. Phosphinothricin N-acetyltransferase Protein, S. viridochromogenes, Recombinant (His & SUMO) is expressed in E. coli expression system with N-6xHis-SUMO tag. The predicted molecular weight is 36.6 kDa and the accession number is Q57146. | |||
TMPY-04218 |
Influenza A H18N11 (A/flat-faced bat/Peru/033/2010) Hemagglutinin/HA Protein (His)
Harvey rat sarcoma viral oncogene homolog |
H18N11 | Baculovirus Insect Cells |
Influenza A H18N11 (A/flat-faced bat/Peru/033/2010) Hemagglutinin/HA Protein (His) is expressed in Baculovirus insect cells with His tag. The predicted molecular weight is 57.7 kDa and the accession number is U5N1D3. | |||
TMPY-00651 |
BACE1 Protein, Human, Recombinant (hFc)
HSPC104,β-site APP-cleaving enzyme 1,ASP2,beta-site APP-clea... |
Human | HEK293 Cells |
BACE1 Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 75 kDa and the accession number is A0A024R3D7. | |||
TMPY-00752 |
BACE1 Protein, Human, Recombinant (His)
β-site APP-cleaving enzyme 1,BACE,beta-site APP-cle... |
Human | HEK293 Cells |
BACE1 Protein, Human, Recombinant (His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 49.9 kDa and the accession number is A0A024R3D7. | |||
TMPY-05546 |
Placental Lactogen/CSH1 Protein, Human, Recombinant (His), Biotinylated
hCS-A,CS-1,CSA,hCS-1,PL,CSMT,chorionic somatomammotropin hor... |
Human | HEK293 Cells |
Placental Lactogen/CSH1 Protein, Human, Recombinant (His), Biotinylated is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 23.7 kDa and the accession number is A8K6C2. | |||
TMPH-00406 |
ctfB Protein, Clostridium acetobutylicum, Recombinant (His & Myc)
Butyrate--acetoacetate CoA-transferase sub... |
Clostridium acetobutylicum | E. coli |
Involved in solventogenic switch which allows C.acetobutylicum to uptake acid and produce solvents. Acts mainly to detoxify the medium by removing the acetate and butyrate excreted earlier in the fermentation. ctfB Protein, Clostridium acetobutylicum, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 30.6 kDa and the accession number is P23673. | |||
TMPH-03078 |
CGTases Protein, Paenibacillus macerans, Recombinant (His)
Cyclodextrin-glycosyltransferase,CGTase,Cyclomaltodextrin gl... |
Bacillus macerans | P. pastoris (Yeast) |
CGTases Protein, Paenibacillus macerans, Recombinant (His) is expressed in yeast with N-6xHis tag. The predicted molecular weight is 13.4 kDa and the accession number is P31835. | |||
TMPH-03583 |
Extracellular elastase Protein, S. epidermidis, Recombinant (His & Myc)
sepA,Extracellular elastase,SEPP1 |
Staphylococcus epidermidis | E. coli |
Protease that has a low substrate specificity. Glucagon is preferentially cleaved between aromatic (Phe) and hydrophobic (Val) amino acids. Hydrolyzes casein and elastin. Extracellular elastase Protein, S. epidermidis, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 37.7 kDa and the accession number is P0C0Q4. | |||
TMPH-00795 |
Glutamate racemase Protein, Helicobacter pylori, Recombinant (His & Myc)
murI,Glutamate racemase |
Helicobacter pylori | E. coli |
Provides the (R)-glutamate required for cell wall biosynthesis. Glutamate racemase Protein, Helicobacter pylori, Recombinant (His & Myc) is expressed in E. coli expression system with N-10xHis and C-Myc tag. The predicted molecular weight is 35.9 kDa and the accession number is B5Z6S2. | |||
------------------------ 更多 ------------------------ |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TMIH-0043 |
3,4-Dihydroxyphenylacetic Acid-d5
|
||
3,4-Dihydroxyphenylacetic Acid-d5 是 3,4-Dihydroxyphenylacetic Acid 的氘代化合物。 | |||
TMIH-0324 |
Medroxyprogesterone 17-Acetate-d3
|
||
Medroxyprogesterone 17-Acetate-d3 是 Medroxyprogesterone 17-Acetate 的氘代化合物。Medroxyprogesterone 17-Acetate 的 CAS 号为 71-58-9。Medroxyprogesterone acetate 是广泛使用的合成类固醇,与雄激素,孕酮及糖皮质激素受体均有作用。 | |||
TMIJ-0025 |
Megestrol Acetate-d3
|
||
Megestrol Acetate-d3 是 Megestrol Acetate 的氘代化合物。Megestrol Acetate 的 CAS 号为 595-33-5。Megestrol acetate 是具有口服活性的合成孕激素。它还具有抗雄激素特性,可用于治疗厌食症和恶病质。 | |||
TMID-0026 |
Acetophenone-d8
|
||
Acetophenone-d8 是 Acetophenone 的氘代化合物。Acetophenone 的 CAS 号为 98-86-2。Acetophenone 是一种有机化合物,能够用作香料。 | |||
TMID-0160 |
5-Hydroxyindole-3-acetic Acid-d6
|
||
5-Hydroxyindole-3-acetic Acid-d6 是 5-Hydroxyindole-3-acetic Acid 的氘代化合物。5-Hydroxyindole-3-acetic Acid 的 CAS 号为 54-16-0。5-Hydroxyindole-3-acetic acid 是 甲氧基肾上腺素或5-羟色胺的主要代谢产物,被用作神经内分泌肿瘤的生物标志物。它是血清素的分解产物,能够从尿液中排出。 | |||
TMID-0261 |
Indole-2,4,5,6,7-d5-3-acetic Acid
|
||
Indole-2,4,5,6,7-d5-3-acetic Acid 是 Indole-3-acetic Acid 的氘代化合物。Indole-3-acetic Acid 的 CAS 号为 87-51-4。3-Indoleacetic acid 是常见的天然植物生长激素。它可以诱导植物细胞的伸长和分裂。 | |||
TMID-0277 |
4-AcetaMido-d3-antipyrine
|
||
4-AcetaMido-d3-antipyrine 是 4-AcetaMido-antipyrine 的氘代化合物。4-AcetaMido-antipyrine 的 CAS 号为 83-15-8。 | |||
TMID-0293 |
Acetylisovaleryltylosin-d3 Tartrate
|
||
Acetylisovaleryltylosin-d3 Tartrate 是 Acetylisovaleryltylosin Tartrate 的氘代化合物。Acetylisovaleryltylosin Tartrate 的 CAS 号为 63428-13-7。Tylvalosin tartrate是一种对革兰氏阳性细菌具有抗性的大环内酯类抗生素。 | |||
TMID-0158 |
Methyl Indole-2,4,5,6,7-d5-3-acetate
|
||
Methyl Indole-2,4,5,6,7-d5-3-acetate 是 Methyl Indole-2,4,5,6,7-3-acetate 的氘代化合物。 | |||
TMIJ-0405 |
2,2,2-Trichloro-acetic Acid-13C2
|
||
2,2,2-Trichloro-acetic Acid-13C2 是 2,2,2-Trichloro-acetic Acid 的 13C 的标记化合物。 | |||
TMIJ-0005 |
Vilanterol-d4 Triphenylacetate
|
||
Vilanterol-d4 Triphenylacetate 是 Vilanterol Triphenylacetate 的氘代化合物。Vilanterol Triphenylacetate 的 CAS 号为 503070-58-4。Vilanterol trifenatate 是一种长效的β2-AR激动剂,效力持续24小时,能够作用于β2-AR (pEC50=10.37),β1-AR (pEC50=6.98) 和 β3-AR (pEC50=7.36)。 | |||
T12447 |
Phenylacetylglutamine-D5
NSC 203800-D5,Phenylacetyl-L-glutamine-D5 |
Others | Others |
Phenylacetylglutamine-D5 is a deuterated form of Phenylacetylglutamine. | |||
TMIH-0090 |
Anthracene-d10
|
||
Anthracene-d10 是 Anthracene 的氘代化合物。 | |||
TMIJ-0168 |
Melitracen-d6 HCl
|
||
Melitracen-d6 HCl 是 Melitracen HCl 的氘代化合物。 | |||
TMIJ-0245 |
Goserelin-d7 Tris-Trifluoroacetate
|
||
Goserelin-d7 Tris-Trifluoroacetate 是 Goserelin Tris-Trifluoroacetate 的氘代化合物。 | |||
TMIJ-0165 |
Glutathione-(glyucine-13C2-15N) Trifluoroacetate
|
||
Glutathione-(glyucine-13C2-15N) Trifluoroacetate 是 Glutathione Trifluoroacetate 的 13C 和 15 N 的标记化合物。 | |||
TMIJ-0404 |
Dibenz[a,h]anthracene-d14
|
||
Dibenz[a,h]anthracene-d14 是 Dibenz[a,h]anthracene 的氘代化合物。Dibenz[a,h]anthracene 的 CAS 号为 53-70-3。Dibenz[a,h]anthracene诱导细菌DNA损伤和基因突变,并在几种哺乳动物细胞培养物中诱导基因突变和转化。 | |||
TMID-0153 |
MELATONIN(ACETYL-d3)
|
||
MELATONIN(ACETYL-d3) 是 MELATONIN 的氘代化合物。MELATONIN 的 CAS 号为 73-31-4。Melatonin 是一种由松果体制成的激素,可激活褪黑激素受体。它在睡眠中起作用,有抗氧化和抗炎特性。它是新型选择性ATF-6抑制剂,可诱导细胞凋亡。 | |||
TMID-0183 |
Flecainide-d4 Acetate
|
||
Flecainide-d4 Acetate 是 Flecainide Acetate 的氘代化合物。Flecainide Acetate 的 CAS 号为 54143-56-5。Flecainide acetate 是位于心脏的 Nav1.5钠离子通道的阻断剂,具有抗心律失常的作用。 | |||
T19442 |
N-acetyl Dapsone (D4')
MADDS D4' |
Others | Others |
N-acetyl Dapsone (D4') is the deuterium-labeled metabolite of Dapsone. | |||
T71145 |
Racecadotril-d5
|
||
Racecadotril-d5 is intended for use as an internal standard for the quantification of racecadotril by GC- or LC-MS. Racecadotril is a prodrug form of the neprilysin (NEP) inhibitor thiorphan. In vivo, racecadotril reduces or prevents castor oil-induced diarrhea without delaying intestinal transit in rats when administered at doses of 80 or 100 mg/kg, respectively. It also decreases the duration of diarrhea and increases body weight gain in a neonatal gnotobiotic pig model of human rotavirus-indu... | |||
T10231 |
Acetazolamide-d3
醋氮酰胺 D3 |
Others | Others |
Acetazolamide D3 is a deuterium-labeled Acetazolamide. Acetazolamide is a potent carbonic anhydrase inhibitor. | |||
TMIH-0087 |
Amlodipine-d4 Maleate (Racemic)
|
||
Amlodipine-d4 Maleate (Racemic) 是 Amlodipine Maleate (Racemic) 的氘代化合物。Amlodipine Maleate (Racemic) 的 CAS 号为 88150-47-4。Amlodipine maleate是一种具有口服活性的二氢吡啶类钙通道阻滞剂,通过阻滞电压依赖性L型钙通道,从而抑制钙离子内流。Amlodipine maleate可用于研究高血压和癌症。 | |||
TMIJ-0046 |
Trimethyl-d9-acetic acid
|
||
Trimethyl-d9-acetic acid 是 Trimethyl-acetic acid 的氘代化合物。Trimethyl-acetic acid 的 CAS 号为 75-98-9。 | |||
TMIJ-0086 |
Acetyl carnitine-d3 HCl
|
||
Acetyl carnitine-d3 HCl 是 Acetyl carnitine HCl 的氘代化合物。 | |||
TMID-0211 |
4-Hydroxyphenylacetic Acid-d6
|
||
4-Hydroxyphenylacetic Acid-d6 是 4-Hydroxyphenylacetic Acid 的氘代化合物。4-Hydroxyphenylacetic Acid 的 CAS 号为 156-38-7。4-Hydroxyphenylacetic acid 是主要的微生物群衍生的多酚代谢物,能够诱导Nrf2表达,具有抗氧化作用。 | |||
TMIJ-0433 |
2,4,5-Trichlorophenoxyacetic Acid-d4
|
||
2,4,5-Trichlorophenoxyacetic Acid-d4 是 2,4,5-Trichlorophenoxyacetic Acid 的氘代化合物。2,4,5-Trichlorophenoxyacetic Acid 的 CAS 号为 93-76-5。 | |||
TMID-0159 |
Indole-3-Acetic-d2 Acid
|
||
Indole-3-Acetic-d2 Acid 是 Indole-3-Acetic Acid 的氘代化合物。Indole-3-Acetic Acid 的 CAS 号为 87-51-4。3-Indoleacetic acid 是常见的天然植物生长激素。它可以诱导植物细胞的伸长和分裂。 | |||
TMID-0101 |
2-Phenylethyl Acetate-d3
|
||
2-Phenylethyl Acetate-d3 是 2-Phenylethyl Acetate 的氘代化合物。2-Phenylethyl Acetate 的 CAS 号为 103-45-7。 | |||
T12693 |
Rasagiline 13C3 mesylate racemic
TVP1012 13C3 racemic,AGN1135 13C3 racemic |
Others | Others |
Rasagiline 13C3 mesylate racemic is the deuterium labeled Rasagiline, which is an irreversible monoamine oxidase inhibitor. | |||
T35515 |
3-Acetyldeoxy Nivalenol-13C17
3-Acetyldeoxy Nivalenol-13C17 |
||
3-Acetyldeoxy nivalenol-13C17is intended for use as an internal standard for the quantification of 3-acetyldeoxy nivalenol by GC- or LC-MS. 3-Acetyldeoxy nivalenol is a mycotoxin that has been found inF. graminearum.1In vivo, 3-acetyldeoxy nivalenol (40 mg/kg) induces duodenal and splenic cell necrosis, as well as lethality (LD50= 70 mg/kg) in mice.2 1.Jiao, F., Kawakami, A., and Nakajima, T.Effects of different carbon sources on trichothecene production and Tri gene expression by Fusarium grami... | |||
T19441 |
N-acetyl Dapsone D4
MADDS D4 |
Others | Others |
N-Acetyl Dapsone D4 is a deuterium-labeled metabolite of N-Acetyl Dapsone, derived from Dapsone. | |||
T10229 |
Acebutolol D7
|
Others | Others |
Acebutolol D7 is a deuterium-labeled Acebutolol. Acebutolol is a selective antagonist of the β1 adrenergic receptor used in the treatment of angina pectoris, hypertension, and cardiac arrhythmias. | |||
TMIH-0071 |
Acetyl L-Carnitine-d3 Chloride
|
||
Acetyl L-Carnitine-d3 Chloride 是 Acetyl L-Carnitine Chloride 的氘代化合物。 | |||
T11036 |
Diacetolol D7
|
Adrenergic Receptor | GPCR/G Protein; Neuroscience |
Diacetolol D7 is deuterium-labeled diacetone Roller. Diacetol is the main metabolite of Acetolol. Diacetololβ-adrenoceptor shielding and anti-arrhythmic agent. | |||
TMID-0057 |
(4-Hydroxy-3-methoxyphenyl)acetic-2,2-d2 Acid
|
||
(4-Hydroxy-3-methoxyphenyl)acetic-2,2-d2 Acid 是 (4-Hydroxy-3-methoxyphenyl)acetic Acid 的氘代化合物。(4-Hydroxy-3-methoxyphenyl)acetic Acid 的 CAS 号为 306-08-1。Homovanillic acid 是一种多巴胺代谢物,它与乳糜泻、生长激素缺乏、芳香族氨基酸脱羧酶缺乏症以及脂联素还原酶缺乏症相关。 | |||
TMIJ-0297 |
Acetylsulfamethoxazole-d4
|
||
Acetylsulfamethoxazole-d4 是 Acetylsulfamethoxazole 的氘代化合物。Acetylsulfamethoxazole 的 CAS 号为 21312-10-7。N4-Acetylsulfamethoxazole 是磺胺甲恶唑的一种代谢物。Sulfamethoxazole 属于磺胺类抗菌素,可用于细菌感染。 | |||
TMID-0304 |
Vitamin A-d5 Acetate
Retinol-d5 Acetate |
||
Vitamin A-d5 Acetate 是 Vitamin A Acetate 的氘代化合物。Vitamin A Acetate 的 CAS 号为 127-47-9。Retinyl acetate 是一种视黄醇的合成乙酸酯形式衍生物,有抗肿瘤和化学预防活性的潜能。 | |||
TMIJ-0318 |
rac-Brivaracetam-d7 (Mixture of Diastereomers)
|
||
rac-Brivaracetam-d7 (Mixture of Diastereomers) 是 rac-Brivaracetam 的氘代化合物。rac-Brivaracetam 的 CAS 号为 357335-87-6。 | |||
T19416 |
Medroxyprogesterone acetate D3
MPA D3,Medroxyprogesterone 17-acetate D3 |
Others | Others |
Medroxyprogesterone acetate D3 is deuterium labeled Medroxyprogesterone acetate. Medroxyprogesterone acetate is a widely used synthetic steroid by its interaction with progesterone, androgen and glucocorticoid receptors. | |||
TMIJ-0039 |
Norethindrone Acetate-2,2,4,6,6,10-d6
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Norethindrone Acetate-2,2,4,6,6,10-d6 是 Norethindrone Acetate 的氘代化合物。Norethindrone Acetate 的 CAS 号为 51-98-9。Norethindrone acetate 是一种雌性激素,对青少年月经和肝腺瘤有抑制作用,常与孕激素联合使用,可用于研究子宫内膜异位症。 | |||
TMIJ-0240 |
Lacosamide-d3 (Acetyl-d3)
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Lacosamide-d3 (Acetyl-d3) 是 Lacosamide 的氘代化合物。Lacosamide 的 CAS 号为 175481-36-4。Lacosamide是一种功能化氨基酸。Lacosamide以一种新的方式调节钠通道:它选择性地增强钠通道缓慢失活,而对快速失活没有影响Lacosamine在不同的啮齿类动物癫痫发作模型中显示出抗癫痫作用,在反映神经性疼痛和慢性炎性疼痛的不同类型和症状的实验动物模型中显示了抗伤害潜力。 | |||
TMIJ-0512 |
Acenaphthene-d10
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Acenaphthene-d10 是 Acenaphthene 的氘代化合物。Acenaphthene 的 CAS 号为 83-32-9。 | |||
TMIJ-0290 |
Acepromazine-d6 maleate
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Acepromazine-d6 maleate 是 Acepromazine maleate 的氘代化合物。Acepromazine maleate 的 CAS 号为 3598-37-6。Acepromazine maleate 是一种 α 肾上腺素受体 (alpha-adrenoceptor) 拮抗剂,是一种吩噻嗪类促进安定的试剂。 | |||
TMIJ-0529 |
Acenaphthylene-d8
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Acenaphthylene-d8 是 Acenaphthylene 的氘代化合物。Acenaphthylene 的 CAS 号为 208-96-8。Acenaphthylene 是多环芳烃。其中多环芳烃是自然衍生于煤和焦油沉积物中,并由有机质的不完全燃烧得到。 | |||
TMIJ-0258 |
Semaglutide-d8 Tetratrifluoroacetate
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Semaglutide-d8 Tetratrifluoroacetate 是 Semaglutide Tetratrifluoroacetate 的氘代化合物。 | |||
TMIJ-0424 |
Chloroacetic Acid-d3
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Chloroacetic Acid-d3 是 Chloroacetic Acid 的氘代化合物。 | |||
TMID-0248 |
Triamcinolone acetonide-d6
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Triamcinolone acetonide-d6 是 Triamcinolone acetonide 的氘代化合物。Triamcinolone acetonide 的 CAS 号为 76-25-5。Triamcinolone acetonide 是皮质类固醇。 它是皮质类固醇激素受体激动剂。 它是抗炎糖皮质激素,局部用于治疗各种皮肤疾病。它的有效性是 prednisone 的八倍。 | |||
TMIJ-0466 |
Acephate-d3 (acetyl-d3)
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Acephate-d3 (acetyl-d3) 是 Acephate 的氘代化合物。Acephate 的 CAS 号为 30560-19-1。Acephate 是能产生胆碱毒性的抗胆碱酯酶杀虫剂。它能够有效抑制蟑螂的AChE,但对大鼠 AChE 的抑制作用较弱。 | |||
TMIJ-0432 |
Sodium Acetate-1-13C
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Sodium Acetate-1-13C 是 Sodium Acetate 的 13C 的标记化合物。Sodium Acetate 的 CAS 号为 127-09-3。Sodium acetate 是常用的实验室试剂。 | |||
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