165
10
8
9
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T37197 |
5-HT1A modulator 2 hydrochloride
|
5-HT Receptor | GPCR/G Protein; Neuroscience |
5-HT1A modulator 2 hydrochloride 是 8-OH-DPAT 的一种衍生物,是5-HT1A 的调节剂,Ki 为 53 nM。 | |||
TQ0311 |
GSK163090
|
Dopamine Receptor; 5-HT Receptor | GPCR/G Protein; Neuroscience |
GSK163090 是选择性和具有口服活性的5-HT1A/1B/1D 受体拮抗剂,pKi 值分别为 9.4、8.5 和 9.7。它抑制血清素再摄取转运蛋白的功能活性,pKi 值为 6.1,具有抗抑郁和抗焦虑活性。 | |||
T0280 |
Spiperone
螺哌隆,Spiroperidol,Spiropitan |
Dopamine Receptor | GPCR/G Protein; Neuroscience |
Spiperone (Spiropitan) 是多巴胺 D2、血清素5-HT1A 和血清素5-HT2A 拮抗剂。它是广泛使用的药理学工具。它具有研究神经系统疾病的潜力。 | |||
T9272 |
Xaliproden hydrochloride
|
Dopamine Receptor; 5-HT Receptor | GPCR/G Protein; Neuroscience |
Xaliproden hydrochloride 是选择性和具有口服活性的5-HT1A 受体激动剂,对大鼠海马中的 5-HT1A 特异性结合位点表现出高亲和力。它也是选择性的多巴胺D2受体拮抗剂,具有抗抑郁和抗焦虑作用,有用于神经退行性疾病的研究潜力。 | |||
T0162 |
Quetiapine
ICI204636,Quetiapin,喹硫平 |
Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor; AChR; Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Quetiapine (ICI204636) 是5-HT 受体激动剂和多巴胺受体拮抗剂,对人5-HT1A 的 pEC50值为 4.77,对人 D2的 pIC50值为 6.33。它用于治疗精神分裂症,以及治疗与 I 型双相情感障碍相关的急性躁狂发作。它对人 D2、HT1、5-HT2A、5-HT2C 受体具有中高等亲和力,pKi 值为 7.25、5.74、7.54和5.55。 | |||
T21011 |
Buspirone
Buspirone free base,Ansial,丁螺环酮 |
5-HT Receptor | GPCR/G Protein; Neuroscience |
Buspirone (Buspirone free base) 是一种azaspiro 化合物,具有抗焦虑药、镇静剂、血清素能激动剂和EC 3.4.21.26(脯氨酸寡肽酶)抑制剂的作用。 | |||
T2132 |
Buspirone hydrochloride
Buspirone HCl,盐酸丁螺环酮,Narol,Buspar |
Dopamine Receptor; 5-HT Receptor | GPCR/G Protein; Neuroscience |
Buspirone hydrochloride (Buspar) 是一种 5HT(1A) 受体激动剂,可用于研究广泛性焦虑症。 | |||
T4560 |
Alprenolol
Alpheprol,阿普洛尔,(RS)-Alprenolol,dl-Alprenolol |
5-HT Receptor; Adrenergic Receptor | GPCR/G Protein; Neuroscience |
Alprenolol (Alpheprol) 是一种非选择性β受体阻滞剂,也是5-HT1A 受体拮抗剂。 | |||
T8593 |
RU 24969 free base
5-methoxy-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole |
5-HT Receptor | GPCR/G Protein; Neuroscience |
RU 24969 (5-methoxy-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole) 是 5-HT1A 和 5-HT1B 受体的选择性激动剂,Ki 值分别为 0.38 和 2.5 nM。它可减少液体消耗并增加向前运动。 | |||
T22236 |
Alprenolol hydrochloride
阿普洛尔盐酸盐,盐酸阿普洛尔 |
5-HT Receptor | GPCR/G Protein; Neuroscience |
Alprenolol hydrochloride 是一种非选择性β受体阻滞剂,也是5-HT1A 受体拮抗剂。 | |||
T6241 |
Quetiapine hemifumarate
Quetiapine Fumarate,ICI-204636,富马酸喹硫平 |
Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor | GPCR/G Protein; Neuroscience |
Quetiapine hemifumarate (ICI-204636) 是5-HT 受体激动剂和多巴胺受体拮抗剂,对人5-HT1A 和人D2的pEC50值分别为 4.77 和 6.33,具有抗抑郁和抗焦虑作用。 | |||
T3046 |
BMY 7378 dihydrochloride
BMY7378 HCl |
Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor | GPCR/G Protein; Neuroscience |
BMY 7378 dihydrochloride (BMY7378 HCl) 是选择性 α1D 肾上腺素受体拮抗剂,也是5-HT1A 受体部分激动剂。它同表达克隆大鼠 α1D-AR 的膜结合的亲和力 (Ki=2 nM) 是同克隆大鼠 α1A-AR (Ki=800 nM) 或仓鼠 α1B-AR (Ki=600 nM) 结合的亲和力 的100 以上。 | |||
T8136 |
Perospirone hydrochloride
Perospirone HCl,盐酸哌罗匹隆,SM-9018 hydrochloride |
Dopamine Receptor; 5-HT Receptor | GPCR/G Protein; Neuroscience |
Perospirone hydrochloride (Perospirone HCl) 是非典型的抗精神病剂,可用于精神分裂症的研究。它是可口服的5-HT2A 受体和多巴胺 D2受体的拮抗剂,也是5-HT1A 受体的部分激动剂。 | |||
T6647 |
Rotigotine-
Neupro,N-0923,罗替戈汀,N-0437,SPM 962 |
Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor | GPCR/G Protein; Neuroscience |
Rotigotine (N-0923) 是多巴胺受体激动剂,是5-HT1A receptor 的部分激动剂,以及α2B-肾上腺素受体的拮抗剂,用于治疗帕金森病和不宁腿综合征。 | |||
T3431 |
Pardoprunox hydrochloride
SLV-308 hydrochloride,DU-126891 hydrochloride,帕多芦诺盐酸盐 |
Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor | GPCR/G Protein; Neuroscience |
Pardoprunox hydrochloride (SLV-308 hydrochloride) 是多巴胺受体 D2、D3部分激动剂和5-HT1A 激动剂,pEC50分别为 8、9.2 和 6.3。 | |||
T0088 |
Urapidil hydrochloride
Urapidil HCl,盐酸乌拉地尔 |
5-HT Receptor; Adrenergic Receptor | GPCR/G Protein; Neuroscience |
Urapidil hydrochloride (Urapidil HCl) 是α1-肾上腺素受体拮抗剂和5-HT1A 受体激动剂。 | |||
T5387 |
LP-211
|
Dopamine Receptor; 5-HT Receptor | GPCR/G Protein; Neuroscience |
LP-211 是一种可透过血脑屏障的选择性5-HT7受体激动剂,Ki 值为 0.58 nM,选择性高于 5-HT1A 受体和 D2受体,Ki 分别为188 和 142 nM。 | |||
T21337 |
Lurasidone
SM-13496,鲁拉西酮 |
Dopamine Receptor; 5-HT Receptor | GPCR/G Protein; Neuroscience |
Lurasidone (SM-13496) 是多巴胺 D2和5-HT7的拮抗剂,IC50值分别为 1.68 和 0.495 nM。它也是5-HT1A 受体的部分激动剂,IC50值为 6.75 nM。 | |||
T1735 |
Lurasidone hydrochloride
Lurasidone HCl,SM-13496 (Hydrochloride),盐酸鲁拉西酮,SM-13496 |
Dopamine Receptor; 5-HT Receptor; Norepinephrine | GPCR/G Protein; Neuroscience |
Lurasidone hydrochloride (Lurasidone HCl) 是多巴胺 D2和5-HT7的拮抗剂,IC50值分别为 1.68 和 0.495 nM,用于治疗精神分裂症和双相情感障碍。它也是5-HT1A 受体的部分激动剂,IC50值为 6.75 nM。 | |||
T4577 |
Cariprazine
卡利拉嗪,RGH-188 |
Dopamine Receptor; 5-HT Receptor | GPCR/G Protein; Neuroscience |
Cariprazine (RGH-188) 是一种新型抗精神病候选药物,结合D3、D2和5-HT1A 的Ki 为0.085、0.49 和 2.6 nM。 | |||
T19917 |
Gepirone
|
5-HT Receptor | GPCR/G Protein; Neuroscience |
Gepirone 属于丁螺环酮家族的 5-HT1A 受体激动剂。它对 5-HT1A 受体的选择性高于 SSRIs。 | |||
T12489L |
Pimethixene maleate
Pimetixene maleate |
Dopamine Receptor; 5-HT Receptor; AChR; Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Pimethixene maleate (Pimetixene maleate) 是一种高效的 5-HT2B 受体拮抗剂,具有镇静和镇咳活性。Pimethixene maleate 抑制 5-HT1A,5-HT2A,5-HT2B,5-HT2C,组胺 H1,多巴胺 D2 和 D4.4 以及毒蕈碱 M1 和 M2,可用于研究儿童干咳和刺激性咳嗽。 | |||
T23285 |
S 14506 hydrochloride
|
5-HT Receptor | GPCR/G Protein; Neuroscience |
S 14506 hydrochloride 是一种5-HT1A 受体完全激动剂。 | |||
T80805 |
WAY-607695
|
5-HT Receptor | GPCR/G Protein; Neuroscience |
WAY-607695 是一种潜在的 5-HT1A 受体激动剂。 | |||
T10168 |
5-HT1A modulator 1
5-HT1Amodulator1 |
Phospholipase; Dopamine Receptor; 5-HT Receptor; Adrenergic Receptor | GPCR/G Protein; Metabolism; Neuroscience |
5-HT1A modulator 1 对 5-HT1A、α1-肾上腺素能受体和 D2 受体具有非常高的亲和力(IC50s = 2 nM、10 nM 和 40 nM)。 | |||
T68172 |
Zalospirone
|
5-HT Receptor | GPCR/G Protein; Neuroscience |
Zalospirone 是一种5-HT1A 受体激动剂,可用于研究焦虑症和重度抑郁症。 | |||
T23007 |
MM 77 dihydrochloride
MM 77二盐酸盐 |
5-HT Receptor | GPCR/G Protein; Neuroscience |
MM 77 dihydrochloride 是一种有效的 5-HT1A 受体突触后拮抗剂,具有抗焦虑样活性。 | |||
T28258 |
Org-13011 fumarate
Org13011,Org 13011 |
5-HT Receptor | GPCR/G Protein; Neuroscience |
Org-13011 fumarate1 是 5-HT1A 受体的激动剂,可用于研究神经系统疾病。 | |||
T23631 |
Adatanserin
WY-50324,WY 50324,WAY SEB 324,WY50324 |
5-HT Receptor | GPCR/G Protein; Neuroscience |
Adatanserin (WY 50324) 是一种混合型 5-HT1A 受体部分激动剂,也是一种 5-HT2A 和 5-HT2C 受体拮抗剂,具有潜在的神经保护活性,可用于研究焦虑和抑郁症。 | |||
T3179 |
Eptapirone
F 11440 |
5-HT Receptor | GPCR/G Protein; Neuroscience |
Eptapirone (F 11440) 是一种高效且选择性的 5-HT1A 受体激动剂,具有显着的抗抑郁和抗焦虑潜力。 | |||
T22379L |
NLX-204 hydrochloride(2170405-10-2 free base)
|
5-HT Receptor | GPCR/G Protein; Neuroscience |
NLX-204 hydrochloride(2170405-10-2 free base)是一种有效且选择性的 ERK1/2 磷酸化偏好 5-HT1A 受体激动剂 (pKi = 10.19)。 | |||
T68059 |
Ebalzotan
NAE 086 |
5-HT Receptor | GPCR/G Protein; Neuroscience |
Ebalzotan (NAE 086) 是一种 5-HT1A receptor激动剂,可用于研究抑郁症。 | |||
T7412 |
Tandospirone citrate
SM-3997 citrate,坦度螺酮柠檬酸盐,枸橼酸坦度螺酮 |
5-HT Receptor | GPCR/G Protein; Neuroscience |
Tandospirone citrate (SM-3997 citrate) 是一种选择性5-HT1A 受体激动剂,Ki 为27 nM。 | |||
T22689 |
CP94253 hydrochloride
CP 94253 hydrochloride |
Others; 5-HT Receptor | GPCR/G Protein; Neuroscience; Others |
CP94253 hydrochloride (CP 94253 hydrochloride) 是一种有效的、特异性的和中枢活性的 5-HT1B 受体激动剂,Ki 为 2 nM。5-HT1A、5-HT1D、5-HT1C 和 5-HT2 的 Ki 分别为 89、49、860 和 1600 nM 。 | |||
T7281 |
F-15599
|
5-HT Receptor | GPCR/G Protein; Neuroscience |
F-15599 是一种高度选择性的 G 蛋白偏向 5-HT1A 受体激动剂,Ki 值为 3.4 nM。 | |||
T0165 |
Urapidil
Mediatensyl,乌拉地尔,Ebrantil,Eupressyl |
5-HT Receptor; Adrenergic Receptor | GPCR/G Protein; Neuroscience |
Urapidil (Ebrantil) 是交感神经抗高血压药物,可作为 5-HT1A 受体激动剂和 α1-肾上腺素受体拮抗剂。 | |||
T61934 |
Repinotan
BAY x 3702 free base |
5-HT Receptor | GPCR/G Protein; Neuroscience |
Repinotan (BAY x 3702 free base) 是一种可透过血脑屏障(BBB)且具有口服活性和选择的 5-HT1A 受体激动剂,具有神经保护活性,可拮抗吗啡诱导的麻醉大鼠通气抑制,可用于研究急性缺血性中风和创伤性脑损伤。 | |||
T16421 |
p-MPPI hydrochloride
|
5-HT Receptor | GPCR/G Protein; Neuroscience |
p-MPPI hydrochloride 是一种选择性的,具有高亲和力的5-HT1A 受体拮抗剂,能穿过血脑屏障,具有抗抑郁和抗焦虑样作用。 | |||
T61816 |
EMD 56551
|
5-HT Receptor | GPCR/G Protein; Neuroscience |
EMD 56551 是一种具有选择性的小分子 5-HT1A 受体激动剂,具有抗焦虑活性,可用于研究焦虑症。 | |||
T24885 |
Tiospirone
BMY 13859-1 |
Dopamine Receptor; 5-HT Receptor | GPCR/G Protein; Neuroscience |
Tiospirone (BMY 13859-1) 是一种 5-HT2 受体拮抗剂,也是一种多巴胺阻滞剂, 抑制 D2,5-HT1a,5-HT7 和 sigma 受体。Tiospirone 可用于研究神经分裂等神经系统相关疾病。 | |||
T1566 |
Aripiprazole
阿立哌唑,OPC-14597 |
5-HT Receptor | GPCR/G Protein; Neuroscience |
Aripiprazole (OPC-14597) 是血清素受体 5-HT1A 和多巴胺 D2 受体的部分激动剂,还用作突触后拮抗剂和血清素受体 5-HT2A 的拮抗剂。 | |||
T71138L |
Binospirone
MDL 73005EF |
5-HT Receptor | GPCR/G Protein; Neuroscience |
Binospirone (MDL 73005EF) 是一种 5-HT1A 受体激动剂,具有抗焦虑活性,可用于研究青光眼和与神经功能障碍相关的运动障碍。 | |||
T2395L |
Vortioxetine hydrobromide
氢溴酸沃替西汀,Vortioxetine (Lu AA21004) HBr,Vortioxetine HBr,盐酸沃替西汀,Lu AA21004 hydrobromide |
5-HT Receptor; Serotonin Transporter | GPCR/G Protein; Neuroscience |
Vortioxetine hydrobromide (Lu AA21004 hydrobromide) 是5-HT1A、5-HT1B、5-HT3A、5-HT7受体和5-羟色胺转运体(SERT)的抑制剂,Ki 值分别为 15、33、3.7、19 和 1.6 nM。 | |||
T27262 |
Enciprazine
WY-48624,D-3112,WY48624,WY 48624,D 3112,D3112 |
5-HT Receptor | GPCR/G Protein; Neuroscience |
Enciprazine (D-3112) 具有抗焦虑活性,对 5-HT1A 受体和 ADRA1有很高的亲和力,可用于治疗焦虑症,可用于研究抑郁症。 | |||
T70044L |
Sarizotan 2HCl
|
5-HT Receptor; HER | Angiogenesis; GPCR/G Protein; JAK/STAT signaling; Neuroscience; Tyrosine Kinase/Adaptors |
Sarizotan 2HCl 是一种 hERG 通道抑制剂和 5-羟色胺5-HT1A受体激动剂,具有潜在的抗抑郁作用,可用于研究帕金森运动障碍。 | |||
T3648 |
Hypidone hydrochloride
YL0919 |
5-HT Receptor | GPCR/G Protein; Neuroscience |
Hypidone hydrochloride (YL0919) 是一种新型抗抑郁候选药物,具有作为 5-HT1A 受体激动剂和选择性 5-羟色胺再摄取抑制剂的双重活性。 | |||
T6423 |
BRL-15572 dihydrochloride
四氢罂粟碱盐酸盐,BRL 15573 dihydrochloride |
5-HT Receptor | GPCR/G Protein; Neuroscience |
BRL-15572 dihydrochloride (BRL 15573 dihydrochloride) 是一种 5-HT1D 受体拮抗剂,pKi 为 7.9,对 5-HT1A 和 5-HT2B 受体也显示出相当大的亲和力,其选择性是 5-HT1B 受体的 60 倍。 | |||
T22871 |
Ipsapirone
|
5-HT Receptor | GPCR/G Protein; Neuroscience |
Ipsapirone 是 5-HT1A 受体的部分激动剂,在高剂量时对 5-HT2 和 α1-肾上腺素能功能产生抑制作用。 | |||
T10249 |
Adoprazine
SLV313 |
Others | Others |
Adoprazine (SLV313) 是 5-HT 1A 受体的完全激动剂,其在 h5-HT1A 受体的 pEC50 为 9。Adoprazine 是 D2 和 D3 受体的完全拮抗剂,在 hD2 受体中的 pA2 值是 9.3,在 hD3 受体中的 pA2 值是 8.9。Adoprazine 具有非典型抗精神病的特征。 | |||
T2631 |
WAY-100635 Monomaleate
|
Dopamine Receptor; 5-HT Receptor | GPCR/G Protein; Neuroscience |
WAY-100635 maleate 是一种选择性的5-hydroxytryptamine 1A 受体拮抗剂,IC50值为 0.91 nM,Ki 值为 0.39 nM。它也是多巴胺 D4受体激动剂,对于5-HT1A 和 α1-肾上腺素的 pIC50值分别为 8.9 和 6.6。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T1045 |
Trimipramine maleate
Surmontil maleate,马来酸三甲丙咪嗪,三甲丙咪嗪马来酸盐 |
Dopamine Receptor; 5-HT Receptor; Antibacterial; Adrenergic Receptor; Norepinephrine; Histamine Receptor | GPCR/G Protein; Immunology/Inflammation; Microbiology/Virology; Neuroscience |
Trimipramine maleate (Surmontil maleate) 是一种 5-HT 受体拮抗剂,对 5-HT1C、5-HT2和 5-HT1A 受体的 pKi 值分别为 6.39、8.10和 4.66。 | |||
T0525 |
Flopropione
夫洛丙酮,Phloropropiophenone |
5-HT Receptor; Transferase | GPCR/G Protein; Metabolism; Neuroscience |
Flopropione (Phloropropiophenone) 是一种解痉剂,用作 5-HT1A 受体拮抗剂,也是儿茶酚-O-甲基转移酶抑制剂。 | |||
T21855 |
AMI-193
Espiramida,螺拉米特,Spiramide |
Dopamine Receptor; 5-HT Receptor | GPCR/G Protein; Neuroscience |
AMI-193 (Spiramide) 是一种有效和选择性的 5-HT2 和 D2 受体,对 5-HT2、D2 受体、5-HT1A、D1 受体和 5-HT1C 受体的 Kis 分别为 2、3、50、2530 和 4300 nM。 AMI-193 显示出抗精神病活性。 | |||
TN1465 |
Cannabigerol
|
NOS; 5-HT Receptor; ROS | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Cannabigerol 是一种植物大麻素,是一种高亲和力 α2-肾上腺素能受体激动剂、中度亲和力 5-HT1A 受体拮抗剂和低亲和力 CB1/CB2受体拮抗剂。它可降低眼压,有潜力治疗青光眼。 | |||
T4429 |
Rauwolscine hydrochloride
Corynanthidine hydrochloride,盐酸育亨宾碱,萝芙素盐酸盐,α-Yohimbine hydrochloride,Isoyohimbine hydrochloride |
Adrenergic Receptor | GPCR/G Protein; Neuroscience |
Rauwolscine hydrochloride (Isoyohimbine hydrochloride) 是一种高选择性的 α2 adrenergic 受体拮抗剂,Ki=12 nM。 | |||
T6648 |
Rotundine
Gindarine,L-Tetrahydropalmatine,Caseanine,罗通定,(-)-Tetrahydropalmatine |
Dopamine Receptor; 5-HT Receptor | GPCR/G Protein; Neuroscience |
Rotundine (Gindarine) 是多巴胺D1、D2和D3受体的拮抗剂,IC50值分别为 166、1.4 和 3.3 μM。 它也是5-HT1A 的拮抗剂,IC50值为 370 nM。 | |||
T2874 |
Tetrahydroberberine
四氢小檗碱,Tetrahydroberberine THB,Canadine |
Dopamine Receptor; 5-HT Receptor | GPCR/G Protein; Neuroscience |
Tetrahydroberberine (Canadine) THB 是一种异喹啉类生物碱,从延胡索中分离得到,对 D2和5-HT1A 受体 uM 级亲和力。 | |||
TN1171 |
6-Dehydrogingerdione
1-Dehydro-6-gingerdione,1-脱氢-6-姜酮 |
NOS; COX; Prostaglandin Receptor | GPCR/G Protein; Immunology/Inflammation; Neuroscience |
1-Dehydro-6-gingerdione is a 5-HT1A receptor partial agonist. | |||
T20647 |
N-Methyllaurotetanine
NSC-247506,NSC247506,Rogersine,Lauroscholtzine,NSC 247506 |
||
N-Methyllaurotetanine is a natural product with good affinity for the 5-HT1A receptor. | |||
TN3393 |
alpha-Yohimbine
|
5-HT Receptor | GPCR/G Protein; Neuroscience |
Alpha-Yohimbine is a 5-HT1A receptor agonist, it is strong selective 2-adrenoceptor antagonist. Alpha-Yohimbine possess aphrodisiac effect. |
Cat. No. | Product Name | Species | Expression System |
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TMPY-05308 |
CD45 Protein, Human, Recombinant (aa 1-529, His)
GP180,B220,L-CA,protein tyrosine phosphatase, receptor |
Human | HEK293 Cells |
CD45 Protein, Human, Recombinant (aa 1-529, His) is expressed in HEK293 mammalian cells with His tag. The predicted molecular weight is 57.4 kDa and the accession number is P08575-5. | |||
TMPY-05387 |
SLAMF7 Protein, Human, Recombinant (hFc)
SLAM family member 7,19A,SLAM7,CS1,CD319,CRACC |
Human | HEK293 Cells |
SLAMF7 Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 49.1 kDa and the accession number is Q9NQ25-5. | |||
TMPY-04318 |
GRIK2 Protein, Human, Recombinant (hFc)
GLUR6,EAA4,MRT6,GLR6,glutamate receptor, ionotropic... |
Human | HEK293 Cells |
GRIK2 (Glutamate Ionotropic Receptor Kainate Type Subunit 2, also known as GluR6) is a Protein Coding gene. The GRIK2 (one of the kainate receptors) gene resides in a genetic linkage region (6q21) associated with bipolar disorder (BPD). The gene coding for GRIK2 has been suggested as a candidate gene for autism based on its localization in the autism-specific region on chromosome 6q21 and the involvement of receptor protein in cognitive functions like learning and memory. GRIK2 belongs to the gl... | |||
TMPY-05547 |
SLAMF7 Protein, Human, Recombinant (hFc), Biotinylated
CS1,SLAM7,CD319,SLAM family member 7,CRACC,19A |
Human | HEK293 Cells |
SLAMF7 Protein, Human, Recombinant (hFc), Biotinylated is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 49.1 kDa and the accession number is Q9NQ25-5. | |||
TMPY-05498 |
SR-BI/SCARB1 Protein, Human, Recombinant (hFc)
HDLQTL6,SR-BI,SRB1,CD36L1,CLA-1,CLA1,scavenger receptor<... |
Human | HEK293 Cells |
SR-BI/SCARB1 Protein, Human, Recombinant (hFc) is expressed in HEK293 mammalian cells with hFc tag. The predicted molecular weight is 73.4 kDa and the accession number is Q8WTV0-5. | |||
TMPJ-00854 |
ETS1 Protein, Human, Recombinant (His)
V-ets Erythroblastosis Virus E26 Oncogene Homolog 1 (Avian),... |
Human | E. coli |
ETS1 Protein (ETS1) is a nuclear protein that belongs to the ETS family. Members of this family recognize the core consensus DNA sequence GGAA/T in target genes. Proteins function either as transcriptional activators or repressors of numerous genes. They are involved in stem cell development, cell senescence and death, and tumorigenesis. ETS1 is a transcription factor, containing one ETS DNA-binding domain and one PNT (pointed) domain. it has been shown to interact with TTRAP, UBE2I and Death As... | |||
TMPK-01357 |
SIRP alpha V5 Protein, Human, Recombinant (His & Avi)
MFR,PTPNS1,P84,BIT,MYD-1,MYD1,SHPS-1,SIRPA,SIRP α,SIRP α V |
Human | HEK293 Cells |
Signal regulatory protein α (SIRPα) is a regulatory membrane glycoprotein from SIRP family expressed mainly by myeloid cells and also by stem cells or neurons.SIRPα acts as inhibitory receptor and interacts with a broadly expressed transmembrane protein CD47 also called the "don´t eat me" signal. | |||
TMPK-01363 |
SIRP alpha V5 Protein, Human, Recombinant (His & Avi), Biotinylated
SIRP alpha,MFR,PTPNS1,SIRP α V5,P84,SHPS-1,BIT,CD17... |
Human | HEK293 Cells |
Signal regulatory protein α (SIRPα) is a regulatory membrane glycoprotein from SIRP family expressed mainly by myeloid cells and also by stem cells or neurons.SIRPα acts as inhibitory receptor and interacts with a broadly expressed transmembrane protein CD47 also called the "don´t eat me" signal.Cancer cells highly expressed CD47 that activate SIRP α and inhibit macrophage-mediated destruction. SIRP alpha V5 Protein, Human, Recombinant (His & Avi), Biotinylated is expressed in HEK293 mammalian c... |
Cat. No. | Product Name | Target | Signaling Pathways |
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T10368 |
Aripiprazole (D8)
OPC-14597 D8 |
Others | Others |
Aripiprazole D8 (OPC-14597 D8) is the deuterium-labeled Aripiprazole. Aripiprazole is a human 5-HT1A receptor partial agonist (Ki: 4.2 nM). | |||
T13300 |
Vilazodone-d8
维拉佐酮D8 |
Others | Others |
Vilazodone D8 is a deuterium-labeled vilazodone. Vilazodone is a combined inhibitor of serotonin specific reuptake (SSRI) and agonist of 5-HT1A receptor partial. | |||
T11295 |
Flibanserin-d4
BIMT-17BS D4,BIMT-17 D4,Flibanserin D4 |
Others | Others |
Flibanserin, a compound identified as BIMT-17, acts as a complete agonist at the serotonin 5-HT1A receptor, with a binding affinity (Ki) of 1 nM, while functioning as an antagonist at the 5-HT2A receptor with a 49 nM affinity. Flibanserin D4 represents a deuterium-labeled version of Flibanserin. | |||
T13308 |
Vortioxetine D8
Lu AA 21004 D8 |
Others | Others |
Vortioxetine D8 is a deuterium labeled Vortioxetine. Vortioxetine is an 5-HT1A, 5-HT1B, 5-HT3A, 5-HT7 receptor and SERT inhibitor (Kis: 15 nM, 33 nM, 3.7 nM, 19 nM and 1.6 nM, respectively). | |||
TMIJ-0112 |
Aripiprazole-d8
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Aripiprazole-d8 是 Aripiprazole 的氘代化合物。Aripiprazole 的 CAS 号为 129722-12-9。Aripiprazole 是血清素受体 5-HT1A 和多巴胺 D2 受体的部分激动剂,还用作突触后拮抗剂和血清素受体 5-HT2A 的拮抗剂。 | |||
TMIH-0314 |
Lurasidone-d8 HCl
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Lurasidone-d8 HCl 是 Lurasidone HCl 的氘代化合物。Lurasidone HCl 的 CAS 号为 367514-88-3。Lurasidone hydrochloride 是多巴胺 D2和5-HT7的拮抗剂,IC50值分别为 1.68 和 0.495 nM,用于治疗精神分裂症和双相情感障碍。它也是5-HT1A受体的部分激动剂,IC50值为 6.75 nM。 | |||
T71211 |
Rizatriptan-d6 benzoate salt
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Rizatriptan-d6 is intended for use as an internal standard for the quantification of rizatriptan by GC- or LC-MS. Rizatriptan is an agonist of the serotonin receptor subtypes 5-HT1B and 5-HT1D. It is selective for 5-HT1B and 5-HT1D receptors over 5-HT1A receptors. Rizatriptan induces vasoconstriction in isolated human middle meningeal arteries. In vivo, rizatriptan reduces head grooming, the number of oculotemporal strokes, eye blinking, and one-eye closures in a Cacna1a mutant transgenic mou... | |||
TMIJ-0242 |
Tandospirone-d8
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Tandospirone-d8 是 Tandospirone 的氘代化合物。Tandospirone 的 CAS 号为 87760-53-0。 | |||
T10681 |
Cariprazine D6
RGH-188 D6 |
Dopamine Receptor | GPCR/G Protein; Neuroscience |
Cariprazine D6 (RGH-188 D6) is a deuterium-labeled Cariprazine. Cariprazine is an antipsychotic agent (D3 receptors, Ki: 0.085 nM; D2 receptors, Ki: 0.49 nM). |