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Targets Recommended: Others

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Cat. No. Product Name Target Signaling Pathways
T37093 4,9-Anhydrotetrodotoxin

4,9-Anhydrotetrodotoxin,4,9-anhydro-TTX

Others Others
4,9-Anhydrotetrodotoxin (4,9-anhydro-TTX) is a derivative of TTX that selectively blocks inward sodium current through Nav1.6 voltage-activated sodium channels (IC50 = 7.8 nM in Xenopus oocytes). [1][2][3] It demonstrates IC50 values of 1.3, 0.34, 0.99, 78.5, 1.3, and >30 &#181M for Nav1.2, Nav1.3, Nav1.4, Nav1.5, Nav1.7, and Nav1.8, respectively.[1]

化合物

4,9-Anhydrotetrodotoxin
Cat.No: T37093
Synonym: 4,9-Anhydrotetrodotoxin,4,9-anhydro-TTX
Target: Others
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