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抑制剂 & 化合物

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同位素标记化合物

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Cat. No. Product Name Target Signaling Pathways
T38613 Tigecycline hydrate

GAR-936 hydrate

Others Others
Tigecycline hydrate (GAR-936 hydrate) is a broad spectrum glycylcycline antibiotic. Tigecycline hydrate is bacteriostatic, that inhibits protein synthesis by binding to the 30S ribosomal subunit of bacteria and thereby blocking entry of Aminoacyl-tRNA into the A site of the ribosome during prokaryotic translation. Tigecycline hydrate is active against resistant strains of Gram-positive and Gram-negative bacteria .
T75279 Tigecycline tetramesylate

Others Others
Tigecycline tetramesylate (GAR-936 tetramesylate)为一款广谱甘氨酰环素类抗生素,对E. coli (MG1655菌株)展现出约125 ng/mL的平均抑制浓度(MIC)。针对Acinetobacter baumannii (A. baumannii)的MIC50与MIC90分别达到1 mg/L与2 mg/L。
T23459 Tigecycline hydrochloride

Others Others
Tigecycline hydrochloride is a first-in-class, broad-spectrum antibiotic. It also has activity against antibiotic-resistant organisms.

化合物

Tigecycline hydrate
Cat.No: T38613
Synonym: GAR-936 hydrate
Target: Others
Tigecycline tetramesylate
Cat.No: T75279
Synonym:
Target: Others
Tigecycline hydrochloride
Cat.No: T23459
Synonym:
Target: Others
Cat. No. Product Name Target Signaling Pathways
TMID-0084 Tigecycline-d9

Tigecycline-d9 是 Tigecycline 的氘代化合物。Tigecycline 的 CAS 号为 220620-09-7。Tigecycline是甘氨酰环素抗生素,对Acinetobacter baumannii(A. baumannii) 的 MIC50和 MIC90分别为 1 和 2 mg/L。它对E. coli(MG1655 菌株) 的平均抑制浓度 (MIC) 约 125 ng/ mL。

同位素标记化合物

Tigecycline-d9
Cat.No: TMID-0084
Synonym:
Target:
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