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抑制剂 & 化合物

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同位素标记化合物

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Cat. No. Product Name Target Signaling Pathways
T15731 Ribociclib succinate hydrate

LEE011 succinate hydrate

CDK Cell Cycle/Checkpoint
Ribociclib succinate hydrate is a highly specific CDK4/6 inhibitor (IC50s: 10 nM and 39 nM, respectively). It also is over 1,000-fold less potent against the cyclin B/CDK1 complex.
T15732 Ribociclib succinate

LEE011 琥珀酸盐,瑞博西尼琥珀酸盐,LEE011 succinate

CDK Cell Cycle/Checkpoint
Ribociclib succinate (LEE011 succinate) 是一种高度特异性的CDK4/6抑制剂,IC50值分别为 10 nM 和 39 nM。它对细胞周期蛋白 B/CDK1 复合物的效力低 1000 倍。
T15730 Ribociclib hydrochloride

LEE011 hydrochloride,瑞博西尼盐酸盐

CDK Cell Cycle/Checkpoint
Ribociclib hydrochloride is a highly specific CDK4/6 inhibitor (IC50: 10 nM and 39 nM, respectively). It is over 1,000-fold less potent against the cyclin B/CDK1 complex.

化合物

Ribociclib succinate hydrate
Cat.No: T15731
Synonym: LEE011 succinate hydrate
Target: CDK
Ribociclib succinate
Cat.No: T15732
Synonym: LEE011 琥珀酸盐,瑞博西尼琥珀酸盐,LEE011 succinate
Target: CDK
Ribociclib hydrochloride
Cat.No: T15730
Synonym: LEE011 hydrochloride,瑞博西尼盐酸盐
Target: CDK
Cat. No. Product Name Target Signaling Pathways
TMID-0003 Ribociclib-d6

Ribociclib-d6 是 Ribociclib 的氘代化合物。Ribociclib 的 CAS 号为 1211441-98-3。Ribociclib (LEE011) 是一种细胞周期蛋白依赖性激酶 CDK4/6 抑制剂 (IC50=10/39 nM),具有特异性和口服活性。Ribociclib 具有抗肿瘤活性,可以阻滞细胞周期,抑制肿瘤细胞增殖。

同位素标记化合物

Ribociclib-d6
Cat.No: TMID-0003
Synonym:
Target:
TargetMol Loading
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