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Search Results for " βamanitin "
Targets Recommended: Others ADC Cytotoxin

3

抑制剂 & 化合物

2

天然产物

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Cat. No. Product Name Target Signaling Pathways
T13474 β-Amanitin

Others; ADC Cytotoxin Antibody-drug Conjugate/ADC Related; Others
β-Amanitin is a cyclic peptide toxin in the poisonous Amanita phalloides mushroom, and inhibits inhibits eukaryotic RNA polymerase II and III. β-Amanitin inhibits protein synthesis.
T74659 Dideoxy-amanitin

Others; ADC Cytotoxin Antibody-drug Conjugate/ADC Related; Others
Dideoxy-amanitin (compound 2) 是一种α-Amanitin 衍生物,是一种强效和选择性的 RNA 聚合酶 II 变结构抑制剂,其 IC50值为 74.2 nM。
T81832 MC-VC-PABC-C6-alpha-Amanitin

Others; Drug-Linker Conjugates for ADC Antibody-drug Conjugate/ADC Related; Others
MC-VC-PABC-C6-alpha-Amanitin是一款针对HER2受体的ADC,包含致癌毒素alpha-Amanitin及单克隆抗体MC-VC-PABC-C6。alpha-Amanitin主要抑制RNA聚合酶IIα。该化合物专一性地靶向HER2阳性肿瘤细胞,主要应用于乳腺癌与胃癌的研究领域。

化合物

β-Amanitin
Cat.No: T13474
Synonym:
Target: Others, ADC Cytotoxin
Dideoxy-amanitin
Cat.No: T74659
Synonym:
Target: Others, ADC Cytotoxin
MC-VC-PABC-C6-alpha-Amanitin
Cat.No: T81832
Synonym:
Target: Others, Drug-Linker Conjugates for ADC
Cat. No. Product Name Target Signaling Pathways
T39562 γ-Amanitin

Others; ADC Cytotoxin Antibody-drug Conjugate/ADC Related; Others
γ-Amanitin an ADC cytotoxin and isolated from the mushroom. γ-Amanitin inhibits RNA polymerase II and disrupts synthesis of mRNA. γ-Amanitin shows similar effects to α-Amanitin and β-Amanitin.
T39649 ε-Amanitin

Others; ADC Cytotoxin Antibody-drug Conjugate/ADC Related; Others
ε-Amanitin is a cyclic peptide obtained from various mushroom species. It exhibits a strong affinity for RNA polymerase II and effectively inhibits its activity.

天然产物

γ-Amanitin
Cat.No: T39562
Synonym:
Target: Others, ADC Cytotoxin
ε-Amanitin
Cat.No: T39649
Synonym:
Target: Others, ADC Cytotoxin
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