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Search Results for " β-adrenergic receptors agonist "

Targets Recommended: Others Adrenergic Receptor

抑制剂 & 化合物

重组蛋白

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Cat. No.	Product Name	Target	Signaling Pathways
T4983	Isoetharine mesylate salt Isoetarine mesilate,异丙肾上腺素甲磺酸盐	Others; Adrenergic Receptor	GPCR/G Protein; Neuroscience; Others
	Isoetharine mesylate salt (Isoetarine mesilate) 是一种 β-肾上腺素能受体激动剂。它还是能够上调 CYP450 表达的孕烷 X 受体(PXR) 激活剂。
T24579	Oxyfedrine L-form HCl Modacor,Oxyfedrine L-form hydrochloride,D563,Ildamen,D 563,D-563	Adrenergic Receptor	GPCR/G Protein; Neuroscience
	Oxyfedrine L-form HCl (Ildamen) 是β肾上腺素受体的部分激动剂，用作冠状动脉血管扩张剂和强心剂。
T25984	(±)-Prenalterol H80/62,H-80/62,H 80/62	Adrenergic Receptor	GPCR/G Protein; Neuroscience
	(±)-Prenalterol (H 80/62) 是一种新的心脏选择性正性肌力化合物，是β-2-和β-1-肾上腺素受体的激动剂，可用于研究慢性充血性心力衰竭。
T14498	Barbadin	Arrestin	GPCR/G Protein
	Barbadin 是一种新型且具有特异性的 β-arrestin/β2-adaptin 相互作用抑制剂，对β-arestin1 的 IC50 值为 19.1 μM，对β-arestin2 的 IC50 值为 15.6 μM。Barbadin 增强氯卡色林对 POMC 神经元和减肥的长期影响，可阻断激动剂促进的原型 β2-肾上腺素能、V2-血管加压素和血管紧张素-II-1 型受体的内吞，可用于研究肥胖。
T30504	BMS-196085 SCHEMBL7042488,BMS196085,CHEMBL322862,FM0D5L3W03	Others	Others
	BMS-196085 is an effective and selective human β( 3) All agonists of adrenergic receptors, in β( 1) Partial agonist activity was 45%.
T68114	nardeterol	Others	Others
	Nardeterol 是β肾上腺素能受体的高亲和力部分激动剂。

化合物

Isoetharine mesylate salt

Cat.No: T4983

Synonym: Isoetarine mesilate,异丙肾上腺素甲磺酸盐

Target: Others, Adrenergic Receptor

Oxyfedrine L-form HCl

Cat.No: T24579

Synonym: Modacor,Oxyfedrine L-form hydrochloride,D563,Ildamen,D 563,D-563

Target: Adrenergic Receptor

(±)-Prenalterol

Cat.No: T25984

Synonym: H80/62,H-80/62,H 80/62

Target: Adrenergic Receptor

Synonym: SCHEMBL7042488,BMS196085,CHEMBL322862,FM0D5L3W03

Species：

Expression System：

Tag：

Cat. No.	Product Name	Species	Expression System
TMPJ-00983	ARRB1 Protein, Human, Recombinant (His) Arrestin β-1,β-Arrestin-1,Beta-Arrestin-1,...	Human	E. coli
	β-Arrestin-1 (ARRB1) is a cytoplasmic protein that belongs to the arrestin family. ARRB1 is expressed at high levels in peripheral blood leukocytes and the central nervous system. ARRB1 regulates agonist-mediated G-protein coupled receptor (GPCR) signaling by mediating both receptor desensitization and resensitization processes. ARRB1 acts as a cofactor in the beta-adrenergic receptor kinase (BARK) mediated desensitization of beta-adrenergic receptors. ARRB1 is believed to play a major role in r...