Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T35834 |
(Sar1)-Angiotensin II
(Sar¹)-Angiotensin II |
||
The substitution with Sar at position 1 of angiotensin II resulted in a partial agonistic activity. | |||
T7575L |
[Sar1, Ile8]-Angiotensin II 3TFA
[Sar1, Ile8]-Angiotensin II 3TFA(37827-06-8(free base)) |
Others | Others |
[Sar1, Ile8]-Angiotensin II 3TFA ([Sar1, Ile8]-Angiotensin II 3TFA (37827-06-8(free base))) 是一种对血管平滑肌具有多种作用的肽。 | |||
T7575L1 |
[Sar1, Ile8]-Angiotensin II acetate
|
RAAS | Endocrinology/Hormones |
[Sar1, Ile8]-Angiotensin II acetate 可激活 NADPH 和 NADH 氧化酶,并刺激血管平滑肌细胞中超氧阴离子的形成。 [Sar1, Ile8]-Angiotensin II acetate 对血管平滑肌有多种作用,包括正常动脉的收缩和培养细胞或病变血管的肥大或增生。 | |||
T7575 |
[Sar1, Ile8]-Angiotensin II
[Sar1, Ile8]-Angiotensin II(3TFA) |
RAAS; Others | Endocrinology/Hormones; Others |
[Sar1, Ile8]-Angiotensin II 是一种在血管平滑肌细胞中有多种作用(如正常动脉的收缩,培养的细胞或病变血管的肥大或增生等)的多肽,。 | |||
TP1224 |
[Sar1, Ile8]-Angiotensin II TFA
Angiotensin 2 TFA,AngiotensinII TFA |
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[Sar1, Ile8]-Angiotensin II (TFA) is a peptide compound that exerts various effects on vascular smooth muscle. These effects include the contraction of normal arteries as well as the hypertrophy or hyperplasia of cultured cells or diseased vessels. | |||
TP1929L1 |
Saralasin acetate(34273-10-4 free base)
|
RAAS | Endocrinology/Hormones |
Saralasin acetate(34273-10-4 free base) 是一种非选择性血管紧张素 II 拮抗剂。 | |||
T76634 |
(Sar1,Ile4,8)-Angiotensin II
|
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(Sar1,Ile4,8)-Angiotensin II是一种对angiotensin II type 1 receptor (AT1R)具有功能选择性的激动剂,能增强胰岛素受体 (IR) 信号和糖原合成,同时还能促进Akt和GSK3α/β的磷酸化,这一过程被胰岛素刺激所增强。 | |||
T75733 |
Saralasin TFA
|
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Saralasin ([Sar1,Ala8] Angiotensin II) TFA,血管紧张素 II (angiotensin II) 的八肽衍生物,作为竞争性血管紧张素 II 受体 (angiotensin II receptor) 拮抗剂,其Ki值达0.32 nM(涵盖74%的结合位点),显示出部分激动剂特性。适应于肾血管性高血压、肾素依赖性(血管紧张素原性)高血压的研究。 | |||
T27229 |
E-4177
E4177 |
Others | Others |
E-4177 is an angiotensin type 1 receptor antagonist. In rat adrenal cortex and liver, E4177 competitively inhibited the specific binding of 125I-[Sar1,Ile8]Ang II, with IC50 being (5.2 +/- 1.0) x 10(-8) M for the adrenal cortex and (1.2 +/- 0.3) x 10(-7) |