Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T22413 |
(R)-Viloxazine Hydrochloride
|
Others; Reductase | Endocrinology/Hormones; Metabolism; Others |
(R)-Viloxazine Hydrochloride是Viloxazine的R型异构体,Viloxazine是一种选择性去甲肾上腺素再摄取抑制剂(NRI),可用作抗抑郁药。 | |||
T60325 |
Viloxazine
Emovit,Viloxazin |
5-HT Receptor; Norepinephrine | GPCR/G Protein; Neuroscience |
Viloxazine (Viloxazin) (Viloxazin) is a dual-action compound that functions as a norepinephrine reuptake inhibitor and exhibits potent agonistic activity towards 5-HT 2C receptors while acting as an antagonist for 5-HT 2B receptors, with respective potency values of EC 50 = 32 μM and IC 50 = 27 μM. Its primary mechanism of action involves the modulation of serotonergic and noradrenergic pathways. Viloxazine is commonly employed in depression research [1] [2]. | |||
T22420 |
(S)-Viloxazine Hydrochloride
(S)-Viloxazine HCl |
Norepinephrine | Neuroscience |
(S)-Viloxazine Hydrochloride 是Viloxazine 的S 异构体。Viloxazine 是一种选择性去甲肾上腺素再摄取抑制剂(NRI),可用作抗抑郁药。 |